Zempilo, Amalungiselelo
"Valium" - na ... Description, uqeqesho, nabalingani isenzo
"Valium" - kungenxa ichiza? na impendulo yalo mbuzo uya kufumana phambili umganyana. We kunixelela nani ngale sixhobo isebenza njani, yintoni iimpawu Lubonakala njengoko kufuneka yaye yintoni zenze ukuba iyafumaneka.
Ifomu kunye nokwakheka zizinto ebekupakishwe
"Valium" - ichiza ukuba zingathengwa ngohlobo ngenaliti, kwakunye iipilisi. Ukuba yinxalenye yale mali?
iqulethe 5 mg diazepam 1 ml isisombululo ngenaliti. Loo medicament ke ithunyelwa 50 okanye 10 ampoules iglasi yobumnyama ml-2, zingafakwa kwiibhokisi kwikhadibhodi.
Ngokuphathelele amacwecwe, zingaqulatha 10 okanye 5 mg diazepam, kodwa izithako zongezelelweyo zilandelayo: umbona starch, anhydrous lactose, calcium stearate, starch pregelatinized, idayi.
Lithetha "Valium" azipilisi zipakishwe iibhokisi zekhadibhodi, leyo iqulathe i Valium Valium.
Pharmacology amachiza
"Valium" - ichiza ebonisa anxiolytic, miorelaksiruyuschee, nadlamkisayo, hypnotics kunye neempawu anti-nokuhlutha izinto.
Ngaphambi kukuxelela ntoni indlela yesenzo imali thina, kufuneka kuqondwe ukuba.
Drug "Valium" unalo igama lokushishina zilandelayo - "Diazepam". Eli chiza fanele ukuba iqela benzodiazepines nokuba ukubaluleka enkulu amayeza.
"Valium" - iyeza ukuba, ngenxa yomsebenzi wayo anxiolytic, nokuphelisa ixhala lwangaphakathi, uloyiko, amaxhala noxinezeleko. Iingcali zithi "Diazepam" yedosi-abaxhomekeke ukusebenza kwinkqubo luvo. Ngamanye amazwi, ngezixa ezincinane (malunga 2-15 mg ngosuku), eli chiza ubangela ekuvuseleleni ukusebenza, kunye (ngaphezu kwama-15 mg ngosuku) - umthomalalisi.
iimpawu imithi
Yintoni ephawulekayo na indlela ngokuthi "Valium"? Action (izihlunu relaxant central) beziyobisi lu dityanisiwe a linyuke ikhaliphe polysynaptic apha emqolo. Ukufumana le ukulungiselela kukhokelela ekuthotyweni uxinzelelo lwegazi, ukwandiswa iimpahla coronary, kwakunye nokuphuculwa ukumelana hypoxia yobuchopho kunye nokwanda umbundu iintlungu.
kinetics
I 'Valium "analogs medicament apho ziboniswa apha ngezantsi, ifunxwe ukusuka iphecana zesisu (ngomlomo). Xa oku ukufakwa kwenzeka ngo-75% kwaye xi ubuninzi ekufikelelwe kuso emva kweeyure 1.5.
Inguqu eziphilayo beziyobisi esibindini. Kule fomu i metabolite esebenzayo kunye nesiqingatha-ubomi. Xa kutyunjwa ichiza ukwenza isiphumo iintsana ekufikelelwe kuso emva kweeyure ezingama-30, yaye abadala, kunye nabantu abadala - ngako 100, kunye iiyure ezingama-48, ngokulandelelana. Kulo mzobo ezimbi zesibindi engapheliyo iintsuku 4.
ukulungiselela kujongwa zivela emzimbeni womntu isikakhulu izintso (90%) ngokohlobo conjugates, kwakunye ayitshintshanga (2%), kunye kunye endleni (8%).
ubungqina
Ziziphi izifo isiguli kunikwa "Valium"? Iingcali Ukubuyekezwa ingxelo ukuba eli chiza luboniswe ukufumana phantsi kwale miqathango ilandelayo:
- ziba izihlunu skeletal kwi azotywe lendawo;
- ukuphazamiseka ixhala;
- myositis, samathambo, bursitis, isinqe-spondylitis samathambo, zihlaselana esinganyangekiyo progressive;
- ngqi;
- lwegazi, ongase, isilonda esiswini kunye duodenum 12 (njengendlela ezongezelelweyo), iposi engabalulekanga;
- ugwayi;
- angina;
- iimeko yiSpasticity, kuquka Cerebral Palsy samathambo kunye kwempixano kwezihlunu skeletal kunye ATHETOSIS;
- etheni iziyobisi;
- syndrome vertebral;
- utywala Nhoza syndrome kunye izinto ezifana nexhala, ukungakhululeki, ukuphazamiseka, lafa;
- isimo epilepticus, ukuphathwa sokuwa;
- izifo zengqondo e zuza kunye nokubeleka (umzekelo, ngxaki kunye sexesheni, gestosis, ukulungiselela abasebenzi);
- nangokhwekhwe kunye nezinye izifo zikhatshwa ukurhawuzelela kunye nochuku;
- isifo Meniere kaThixo ;
- karhulumente hallucinatory-paranoid, motor excitation of imvelaphi ezahlukeneyo (in zengqondo kunye yeenkqubo zengqondo);
- zomzimba jikelele kunye premedication (umzekelo, phambi utyando kunye neenkqubo endoscopic).
Izimo
Xa kufuneka usebenzise eli chiza njenge "Valium '? Isiphumo sale ichiza akufani singathanda, ukuba ukuyamkela:
- ku hypersensitivity;
- isiqaqa, ukothuka;
- ukunxila okanye utywala olunamandla;
- iindlela zale izifo esibindini;
- myasthenia gravis;
- engile-ukuvalwa glaucoma;
- kubantwana abancinane ngaphezu kweenyanga ezi-6;
- ngexesha zisanyisa, kwaye kwithuba leenyanga ezintathu yokuqala yokukhulelwa.
Ichiza "Valium": imiyalelo yokusebenzisa
Nikezela ingqalelo indlela kufuneka liyincutshe onamava kuphela. Izigulane abadala umthamo we ichiza emva Ulawulo ngomlomo kufuneka 5-20 mg ngosuku. Le mfumba ichiza kumiselwa ngokuxhomekeke ubukhali iimpawu zesifo, kwakunye umfanekiso clinical iyonke.
Olona nyango iphezulu ithamo kunokwenzeka ayikho ngaphezu kwe-10 mg. Ikhosi therapy oku kuthetha kwimeko ukuphazamiseka ixhala kufuneka liqhubeke 6 iiveki. Emva kweli thuba kufuneka ujonge kugqirha kokuya, kangangokuba wathabatha idosi yesondlo ubuncinane.
Ukupheliswa ichiza ngcembe ingqalelo.
Kwiimeko ezingxamisekileyo, medicament esebenzayo kwazo parenterally (intramuscularly okanye yegazi). Kulo mzekelo, umthamo we 2-20 mg.
Kunye nokubandakanywa efakwa ye ichiza kufuneka ufakwe kancinci, ngeqondo elingagqithanga ml 0.5-1 ngomzuzu.
imiphumela emibi
Njengayo nayiphi na amayeza, ukuthatha phantsi ingqalelo ichiza kunokubangela ukusabela. Ezi ziquka oku kulandelayo:
- bradycardia okanye hypotension;
- kunciphisa ingqondo kunye neqondo asabela;
- ukuba likhoboka leziyobisi;
- isiyezi kunye intloko ebuhlungu;
- uphuhliso ngayo ngamazwi ixhala, sokulibala, nemibono, nokuxutha;
- imemori yokuthothisa (short);
- reactions yokwayama kuyo inaliti;
- nengxaki intshukumo efana dysarthria kunye Ataxia;
- umonakalo nezintso nomhlehlo wesibindi, amathumbu atony, sinciphise yobuntu kunye amandla (ukusetyenziswa ixesha elide ichiza);
- ziyabagulisa;
- syndrome yokuyeka;
- lehla ukusebenza, kunye buthathaka kwezihlunu.
Ekuqeshweni ichiza kwisigulana kubaluleke kakhulu ukwazisa ukuba eli chiza. Emva njengento eyaziwa arhente psychotropic tranquilizer, nto leyo iba inani iziphumo ezibi, phakathi kwazo ingakumbi wachacha iziyobisi kunye ukurhoxiswa.
Dr. Ekumiseleni eli yeza unyanzelekile ukuba ukwazisa isigulana malunga imiphumela emibi ichiza emzimbeni wakhe, kwakunye nokubonelela ezinye iindlela zonyango.
libanda, yamayeza
Overdosing ingqalelo indlela ezingemnandi ephelekwa iimpawu ezifana CNS kukudakumba. A meko efanayo, lungathi lube ezahlukahlukeneyo elihlabayo, ukusukela ukozela kunye nesiphelo isiqaqa. Kwakhona, xa uthatha ngeedosi eziphezulu beziyobisi hypotension kunokwenzeka yesigulane, ukudideka kunye nokudandatheka zokuphefumla.
Unyango kweemeko ezinjalo kunye kunciphiso, ukuba isigulane lisezingqondweni na, iquka uqhelwaniso emesis kunye nokusetyenziswa carbon yasebenza. Xa kunjalo, ukuba isigulana zingqondweni, ukuba ndizihlambile ngokusebenzisa olumayelana isisu, kwakunye unyango kwangumqondiso, ukuvavanyela imisebenzi ebalulekileyo kunye nokuqaliswa ulwelo ukwandisa diuresis.
Ukuze sibophe ukuphazamiseka ngokugqithisileyo isigulane, unganika ngayo barbiturates.
Intsebenziswano kunye nezinye iindlela zonyango
Le medicament "Valium" ebangela potentiation yeziphumo utywala, hypnotics, anticonvulsants, iiarhente iqinile kunye antihistamines, kunye antipsychotics, iintlungu jikelele, lakhula tricyclic, relaxants kwezihlunu kunye analgesics.
evuselela Analeptic kwaye kakhulu ukunciphisa umsebenzi "Diazepam" iziyobisi.
Asidi ukunciphisa umlinganiselo, kodwa hayi inqanaba kukufakwa ichiza.
inhibitors ezifana of microsomal igcwala njenge "Cimetidine", "Omeprazole" "ketoconazole" "fluoxetine" yaye "Fluvoxamine" lokutshintsha pharmacokinetics beziyobisi phantsi ingqalelo, kwaye kananjalo kwandisa ixesha neziphumo zalo zonyango.
"Rifampicin" kunciphisa uyondelelwano lwee- "Diazepam 'igazi, yaye" Erythromycin "imenza yokucolwa layo esibindini.
amachiza afanayo
Yintoni indawo le neziyobisi "Valium '? Analogue eRussia Abathengiswa ezikhemisti. Ngaphezu koko, la machiza zikhutshwa kuphela emva ntetho lokumiselwa zonyango.
Buyisela akakwazi "sibazon", "diazepam" okanye "Diapamom" iziyobisi. Nangona kunjalo, oku kufuneka kwenziwe kuphela emva kokubonisana nogqirha.
Iindleko ichiza
Njengoko kukhankanyiwe ngasentla, ukuthenga iziyobisi "Valium Roche" eRashiya akakwazi kuzo zonke ekhemesti. Iindleko ichiza - malunga liwaka engange (pack ngalinye).
Ixabiso lemali kwi UK kunye namanye amazwe aseYurophu, ngokuqhelekileyo malunga amabini anamashumi amahlanu eemina nganye amacwecwe amawaka (10 mg).
Ukuze ukuthenga kuloo mzi enjalo ichiza eliya kudibana nazo zonke iimfuno nokhuseleko kunye nomgangatho, iingcali Siyaleza isicelo imvelaphi, apho uya kunikwa inkcazelo epheleleyo malunga nokufumaneka kwayo ezikhemisti kunye namaxabiso nenzuzo.
ncomo Consumer malunga namayeza
"Valium" - kuthandwa kakhulu phakathi izigulane ichiza esetyenziswa njenge anxiolytic, miorelaksiruyuschego, nadlamkisayo, hypnotics, kunye anticonvulsants. Ngokutsho impendulo uninzi yabathengi, uthathwa amayeza kakuhle kakhulu ukwenzela izifo ezahlukahlukeneyo, kuquka isifo sokuwa, zokulala, ixhala njalo njalo. Kwakhona ukuthatha kuyanceda lula iimpawu njengoko kukuphazamiseka, lafa nokuphelisa nemibono.
Nangona kunjalo, akukho isixhobo yokuba wayeza alunakulungela wonke ubani. Abanye abantu abasebenzisa eli chiza awonwabanga. Bakuphawula abanikaziyo ukuba ichiza aqale ukwenza kuphela emva kweveki. Ukongeza, kunye nokusetyenziswa ukuqhubekeka medicament kubangela inani elikhulu reactions cala kwaye ikhokelela likhoboka lazo.
Similar articles
Trending Now