ZempiloAmalungiselelo

Ichiza "Ondansetron": analogue, imiyalelo ukusetyenziswa, ixabiso

Kukho ezimbi ezininzi efuna ukufumana antiemetics, ukuvumela ukususa isicaphucaphu kunye neempawu yityhefu. Oku kubaluleke ngakumbi kwixesha postoperative, xa umzimba esuka zomzimba. Kufuneka kwakhona ukuba imiselwe ichiza ngexesha ichemotherapy kunye nonyango radiation. Ezi ziquka iindlela ezisebenzayo ukunyanga "Ondansetron". Analogs ( "Emetron" iziyobisi "Latran" "Zofran") kwaye ngexesha elifutshane ziya ukususa iimpawu kunxilwe kunye nokugabha.

amayeza Action "Ondansetron"

Amayeza fanele ukuba iqela antiemetics. Eyiyo ngexesha elifutshane, kuwukhulula isicaphucaphu nokugabha, owenzeka kwixesha postoperative emva ichemotherapy kunye radiotherapy. Isiphumo ichiza kukuba zinokuyithintela ngokukhetha serotonin 5-HT3 receptor. Ngenxa nokuncipha le reflex gag.

Emva arhente sokungenisa ako ngokukhawuleza esiswini. Phantse 100% enxulumene iiproteni igazi. Isibindi bangenwe ukutya eliphezulu. Zingaphelanga iiyure ezine ichiza ifikelela ifuthe layo ezinintsi nezinyangayo. Phe isicaphucaphu nokugabha ngenxa medicament "Ondansetron". Analogs nawethutyana, imithi iipropati ezifanayo kwaye endaweni ngokupheleleyo yokuqala.

Iimpawu kunye Izimo

The main izinto ezibonisa - unyango kunye nothintelo isicaphucaphu nokugabha emva ichemotherapy kunye radiotherapy, ngokunjalo kwisithuba postoperative. Kukho ezinye Izimo:

  • Awukwazi ukuthatha iyeza kwisiqingatha sokuqala yokukhulelwa;
  • hypersensitivity ukuba amacandelo;
  • zilawulwa ngokuqaphela ukuba izigulane isifo sezintso zesibindi.

isicelo

Ichiza unikwa qho ngamnye. yangosuku kuxhomekeke ubungqongqo iimpawu, kunye ukunxila ngokugqithisa radiation kunye nechemotherapy. Kweli xesha emva kokuba amayeza umsebenzi onikwe izihlandlo eziliqela ngemini de Ukunyamalala ngokupheleleyo iimpawu isicaphucaphu nokugabha. ugqirha kuphela ukumisela njengendlela "Ondansetron» (Ondansetron). Imiyalelo ukuba ichiza ngaphakathi kwikhava ekhemesti.

Akunconywa co-lezolawulo inducers kwinkqubo cytochrome enzymatic, nto leyo enokukhokelela ukuhla kugqitywe kunye nokunyamezelana ukwimo engundoqo (ondansetron).

Akwenzeki ukuba ukumisela ichiza kwithuba leenyanga ezintathu yokuqala yokukhulelwa. Ukuba ufuna ukusebenzisa iziyobisi ngexesha zisanyisa, kuyimfuneko ukuba bayeke ukutya. Kwakhona izigulane emva kotyando esiswini kufuneka uthathe ichiza ngobunono ukwenzela ukuba ukufihla iimpawu kwimiqobo ahlekise emathunjini. Ekubeni isifo sesibindi ayikwazi ngaphezu 8 mg ithamo medicament "Ondansetron".

Analogs nokubonakaliswa amaxabiso Izimo - yonke le nkcazelo kuyimfuneko ukuba ukhankanye phambi unyango.

Ixabiso ichiza - malunga $ 100 isiqwenga nganye.

kahle imithi:

  • intloko;
  • ezayo umbono awucaci kunye nesiyezi;
  • zokucutha;
  • tachycardia;
  • ziyabagulisa;
  • komzimba eshushu intloko yam.

"Latran"

Libhekisela antiemetics. Ngempumelelo kuwukhulula iimpawu isicaphucaphu nokugabha kwixesha postoperative, ngethuba labe radiotherapy. Ichiza ekwaziyo evalela i serotonin uyakhetha receptors-5-HT3. Xa ukuginyile, amayeza ixesha elifutshane wendele esiswini. Phantse 100% enxulumene iiproteni igazi. Pass yokucolwa esibindini yi hydroxylation.

Ukufumaneka benani ichiza iyazalisekiswa iiyure ezine yokuthatha kwedosi yokuqala. Isenzo esinjalo okukuchaphazela amayeza komzimba "Latran". It has a arhente ipropati efanayo "Ondansetron". Analogue, ntonye kunye neziyobisi generic zinokusetyenziswa kuphela emva kothetha-thethwano kunye nogqirha wakho.

Iindleko imithi 180-200 engange ezikhemisti ezahlukeneyo.

Iimpawu ze isicelo

Uthintelo kunye nonyango lwe isicaphucaphu nokugabha kwixesha postoperative, yaye emva ichemotherapy kunye radiotherapy. Awukwazi ukwabela arhente kwithuba leenyanga ezintathu zokuqala zokukhulelwa kunye kwimeko hypersensitivity ukuya ichiza. Kwakhona, akukho indlela emiselwe ngezifo kwesibindi kunye nezintso. Ichiza ayikwazi ingasetyenziswa ukonakalisa ukutya okanye utywala.

Iidosi lusekiwe qho ngamnye kwaye kuthathelwe ingqalelo nobungozi besi sifo. Le khosi ixhomekeke iimpawu kunye ebusweni ukunxila eziphilayo. Umntu akanako ukuthatha libambisene emacwecweni, ezo inhibitors of cytochrome isozyme. Ngaphandle kokubonisana ugqirha ayikhuthazwa ukuba ichiza "Latran", kwakunye nesixhobo sonyango "Ondansetron" (Solution for inaliti). Le miyalelo achaza indlela yokusebenzisa amayeza kuphela iinjongo zokunika ulwazi.

imiphumela emibi

Kwiimeko ezininzi, ichiza laye ukunyamezeleka kakuhle. Ezi mpawu zilandelayo kwenzeka kunqabile kakhulu:

  • ukungaboni kunye nesiyezi, ukuze idlule;
  • intloko ebuhlungu;
  • bradycardia;
  • ukuhla okubonakalayo uxinzelelo;
  • nokuqunjelwa;
  • walunywa;
  • kuyabuya ubushushu.

Awukwazi ukwabela isisombululo okanye icwecwe ngexesha yokumitha zisanyisa. Kwakhona, isilumkiso kufuneka imiselwe emva kotyando phezu peritoneum, ukuze ukuphoswa iimpawu kwimiqobo ahlekise emathunjini. La manyathelo ekufuneka ilandelwe unyango "Ondansetron" iziyobisi. Imiyalelo yokusebenzisa, analogs, idosi echanekileyo - zonke iinkcukacha kufuneka ifundwe phambi kuthomalaliso, yaye ukuba unayo nayiphi na imibuzo zibhekisela oyingcali icebiso.

"Zofran"

Agent ibhekisa kwiqela antiemetics. Ngempumelelo kuwukhulula iimpawu isicaphucaphu nokugabha ngexesha ichemotherapy, kunye nonyango radiation emva kotyando. Iindlela unokukhetha ukuvala serotonin receptors-5-HT3, nto leyo kunciphisa uphawu yityhefu. Phantse 100% enxulumene kwiiproteni igazi. bioavailability obukhulu waphawula emva kweeyure-4 emva ukuthatha iyeza. In "Zofran" oko ikakhulu umzimba esibindini ubuncwane eziphambili izibonelelo zonyango. Pre kufuneka kufundwa phambi kokuba usebenzise amachiza "Ondansetron" umyalelo. Analogs uqobo musa zahluke kumafa nokubonakaliswa. Ngaba "Zofran" malunga 300 engange.

ukusebenzisa Iimpawu

Eyabelwe ngonyango kunye nothintelo elithile lithatha ixesha emva kotyando kunye ichemotherapy kunye nonyango radiation. Kufuneka kuthathwe kwisiqingatha sokuqala zokukhulelwa kunye ngethuba lokuncancisa. Kwakhona akucetyiswa xa kwimeko hypersensitivity ukuya ichiza. Le medicament ingasetyenziswa ukunqanda iimpawu ukugabha kunye nokurhoxiswa ngexesha ukunxila ityhefu.

Umthamo imisela kuphela ngugqirha, kwaye oko kuxhomekeke ebukhulwini isigulane emva labe nasemva utyando. Ichiza kuthathwa ukugqibezela Ukunyamalala iimpawu ukunxila. Akukhuthazwa ukuba co-lezolawulo inhibitors benkqubo isoenzyme isochrome. Oku kufuneka kuqwalaselwa unyango "Ondansetron" iziyobisi. analogue Drug ngokupheleleyo nako ukubuyisela original usindise emikhuhlaneni ukugabha isicaphucaphu.

kahle imithi:

  • ezayo isiyezi kunye ukungaboni;
  • intloko ebuhlungu;
  • kwesisu okanye ukurhuda;
  • hliswa wegazi;
  • bradycardia;
  • intlungu esiswini.

Xa elivela kuzo naziphi na iimpawu ezigatya kufuneka bafune iingcebiso zonyango. Ingcali ukunciphisa idosi okanye ukunika indawo esemgangathweni.

"Emetron"

amachiza Antiemetic ukuba asithe receptors serotonin kwaye kunempembelelo engundoqo.

Iyeza yenziwe ngohlobo kwesisombululo olutyheli kunye namacwecwe. Iimali ezenzelwe ngokupheliswa ukugabha kunye isicaphucaphu emva kutyando ngexesha ichemotherapy kunye radiation therapy. Kuba ulawulo intramuscular okanye efakwa, waphawula ukusebenza kunye nokuncipha zinetyhefu imizuzu eli-10. Isiphumo efanayo "Ondansetron" solution ukulungiselela. Analogue ziyafana kakhulu kumafa.

Ixabiso beziyobisi kwiikhemesti ngaphezulu engange 1,200 pack nganye.

Iimpawu kunye Izimo

Lwanziwa ukuphelisa isicaphucaphu nokugabha ngexesha kutyando ngexesha ichemotherapy kunye radiation therapy abantwana kunye nabantu abadala. asinakusetyenziswa ukuphelisa ukunxila kweziyobisi kwimeko yityhefu. Kukho Izimo ezininzi:

  • ngexesha lokukhulelwa;
  • zisanyisa;
  • ukuya kwiminyaka-2;
  • hypersensitivity yecandelo esebenzayo.

Ichiza yayisalawulwa ne nedosi ye-mg 8 ukuya 32 ngosuku. yangosuku kuxhomekeke ebukhulwini ukunxila kunye neempawu ngabanye eziphilayo. Amanyathelo eyabelwe izigulane unyango kunye ngezifo kwesibindi kunye nezintso. Kwakhona lithetha "Emetron" ngeedosi ephantsi ezisetyenziswa abadala.

reviews

Kwiimeko ezininzi, ichiza unalo ingxelo eyakhayo kwaye zivunwe kakuhle zizigulane. Ekuhambeni kwexesha elifutshane isusa iimpawu ukunxila, kubangele ukugabha kunye isicaphucaphu. Iyeza akubangi umonakalo emzimbeni kwaye kwenziwa ukuya yokuduka ngokupheleleyo iimpawu yityhefu. Ngokutsho iimpendulo ezigulane kunye oogqirha bakwazi ukuphuhlisa i uxabane ukuba ichiza "Ondansetron". Analogue kwemali angangunobangela wokuhlaselwa ezindlwini zazo kunye nokothuka anaphylactic. Ngoko oyidlayo iiseti kuphela ingcaphephe kuthathelwa ingqalelo iimpawu ngamnye malunga nesigulane eso.

Ichiza ayikhobokisi kwaye alahlwa ngokohlobo amacwecwe kunye nesisombululo, nto leyo efanelekileyo nasiphi na isigulane kunye nenkqubo ubungnqongqo. imixube ezinjalo ingasetyenziswa nge kwiminyaka emibini ubudala. Thenga namayeza na ekhemesti. Oogqirha abaninzi bancome iyeza ukuze bawubuyise iimpawu ukunxila.

Ukuba kukho imfuneko yokuba amisele isixhobo ngexesha lokuncancisa, kuhle ukushiya zisanyisa. Iingcali qaphela ukuba isithako esebenzayo ungena ubisi kwaye kwenzakalisa impilo usana. Kakade ke, njengoko phambi kokuthatha naliphi na ichiza kufuna ngokudlana logqirha - ngoko umngcipheko yeziphumo ebezingalindelekanga iza kuncitshiswe.

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