Zempilo, Amalungiselelo
Tablets "Lenuksin": ncomo, imiyalelo ukusetyenziswa, inkcazo, analogue, ixabiso
Indlela zokumelana nokungonwabi ngokwabo? Phendula lo mbuzo kunzima kakhulu. Ngapha koko, ukuba uphume kule karhulumente ngaphandle koncedo lweengcali iyakwazi ezimbalwa. Kule meko, sicebisa ukuba udibane nogqirha, owathi kamva amisiweyo unyango olusebenzayo.
ulwazi jikelele
Ukudakumba kuthiwa ukuphazamiseka kwengqondo, nto leyo luphawulwa imo ephantsi, wacinga disorder (longanyelwe nembono ophambene yonke into eyenzekayo, imigwebo ezimbi, njalo njalo.), Motor abazizidalwa, kwakunye ukulahleka ubuchule ukuba uvuyo.
Kufuneka kuqatshelwe ukuba kule meko, umntu uvikivwa ukuzithemba, yalahleka umdla ebomini kunye nomsebenzi. Kwiimeko ezininzi, isigulana umntu oxinezelekileyo angaqalisa ukukuxhaphaza iziselo ezinxilisayo, Narcotics kunye namanye amachiza psychotropic. Amaxesha amaninzi aba bantu sinotyekelo ukuzibulala.
Namhlanje, ukudakumba ngcono. Kwinkqubo kwezinto psychotropic linokwenziwa ukuba kwanonyango nomonde. Zibhale kakhulu kakhulu. Kungenxa yoko le nto kufuneka amisele liyincutshe onamava kuphela.
bucala
Iyeza ithandwa kakhulu ngenxa yokugula ngengqondo yi yeQela "Lenuksin". Kweli nqaku, siza kukuxelela malunga iimeko apho yena nguye omisiweyo, ukuba unazo naziphi na Izimo kunye neziphumo ebezingalindelekanga, yaye yintoni na ixabiso layo, ifomu ukukhululwa, isakhiwo, nokuba kukho analogue of medikmenta njalo-njalo.
Ukubunjwa ichiza, zempahla epakishwayo nokumila
Phambi ndithi kuni ngendlela amayeza "Lenuksin" izenzo, nto leyo ncomo uya thaca apha ngasezantsi, kufuneka inike uhlobo ukukhululwa. Esi sixhobo kuthengiswa ngohlobo tablets, apho isale yayisoma film.
Ichiza iqulathe icandelo esebenzayo ezifana escitalopram oxalate. Ngaphandle kulo, emacwecweni kunye nezinto abancedisayo ke ngokohlobo microcrystalline kwincindi, isodiyam croscarmellose, talc, microcrystalline neselulosi silitsinizirovannoy, siliconized microcrystalline neselulosi nezinki stearate.
Drug "Lenuksin", nto leyo kunokuba ixabiso eliphezulu, kuthengiswa ezineengqayi ezinepolypropylene (mhlawumbi e namadyungudyungu), sibekwe ngendlela ibhokisi. Umphanda ngamnye iqulethe tablets 28 okanye 14.
Ezona mpawu imithi ye yeQela
Drug "Lenuksin", ukubuyekeza apho ezingaphezu kwe-HIV, i yeQela. Le SSRIs, nto leyo eyandisa xi le neurotransmitters emqhokrweni zobuchopho, kwaye tsala kwaye iphucula ukusebenza ngomhla receptors serotonin postsynaptic.
ifana isiqalelo medicament ngoku ukubophelela Alpha-adrenoceptors, m-cholinergic receptors, opioid, serotonin, benzodiazepine, dopamine nezamkeli histamine.
Practice ibonisa ukuba isiphumo bucala kwizigulane iqala ukuphuhlisa iiveki kuphela emva 2-4 emva unyango. Le intlawulo iphezulu sisiphumo of one- kudla kwafezekiswa isibini kweenyanga.
Pharmacokinetics kuthetha
Njengoko ichiza ako, "Lenuksin"? ngokusetyenziswa manual bucala ithi nokufunxwa yayo ezimeleyo ekudleni. Le bioavailability ye ichiza nama-80%. Xi igazi liphezulu kufikelelwa emva kweeyure 4 ex. medicament Plasma protein esibophelelayo nama-56%.
nethe bucala kwenzeka esibindini (ukwenza didemetilirovannyh esebenzayo kunye metabolites demethylated). Kwisiqingatha ubomi emva kulawulo ezininzi nama-30 iiyure.
Iimpawu zibonisa ukuba ukusetyenziswa noxinezeleko
Kwezinye iimeko, ichiza "Lenuksin"? Imiyalelo yokusebenzisa, iimpendulo zibonisa ukuba kufuneka isetyenziswe kuphela phantsi zokwahluka zilandelayo:
- ukudakumba, kuba uhlobo kakhulu okanye ulungise;
- Social ixhala disorder (lumo leyo);
- ukuphaphazela disorder ne agoraphobia, okanye ngaphandle kwayo;
- ngokubanzi nexhala disorder.
Izimo ukusetyenziswa yokunciphisa
Treatment kunye lakhula kuyo nayiphi na imeko kwenziwa phantsi kwale miqathango kunye zinto zilandelayo:
- ngokuthi utye ngaxeshanye Mao inhibitor;
- e esakhula ukuya kwiminyaka eli-18;
- hypersensitivity ukuya medicament okanye iinxalenye zayo;
- kusilela okanye isomaltase sucrase, iswekile-galactose malabsorption kunye fructose ukunganyamezelani.
ukusebenzisa ukuqapha
Tablets "Lenuksin" kufuneka inikwe izigulane ukusilela kwezintso na ngononophelo kakhulu, isifo seswekile, hypomania, ukopha ukuthambekela, mkhuba, ukuqina kunye ukuxhuzula pharmacologically olungalawulwayo.
Kwakhona kufuneka ngenyameko kakhulu ukuba ukusebenzisa le iyeza nokudakumba kunye notyekelo ukuzibulala, ngoxa ukufumana amachiza ukwehlisa embundwini kwaye umzimba isoenzymes ka CYP2C19, abadala, kunye ne-ethanol.
Drug "Lenuksin": imiyalelo yokusebenzisa
Eli chiza ngesi ekhemesti ngokumiselwa kuphela. Ngapha koko, oko kumisela kuphela iingcali abaye izifundo eziyimfuneko.
Le umthamo ichiza kunye ubuninzi kwayo ukusetyenziswa ixhomekeke kubungakanani kunye nohlobo kutenxa kokumiselweyo. Ngokutsho umyalelo, wathi iindlela kufuneka zisetyenziswe kanye ngosuku, phambi, emva, okanye phakathi izidlo.
- Depression, ukuba ubume enzima okanye avareji.
Kulo mzekelo, ichiza "Lenuksin", nto leyo kunokuba ixabiso eliphezulu abizwa i-10 mg kanye ngemini. Kuxhomekeka abasabela ngayo (ngamnye) yomguli, idosi kufuneka kwandiswe ukuze mg-20 ngosuku. Emva yokuduka iimpawu zokudakumba kufuneka baqhubeke unyango iinyanga ezi-6, ukulungisa isiphumo.
- One- ne agoraphobia, okanye ngaphandle kwayo.
Kulaa veki yokuqala yonyango isigulane efunekayo ithamo esilingana 5 mg ngosuku. Kwixesha elizayo kufuneka kwandiswe kanye kabini. Kuxhomekeka isixa abasabela ngayo ichiza isigulane nga kusondela kuwo ubuninzi, ngamanye ku-20 mg ngosuku. Le unyango ihlala iinyanga eziliqela.
- lumo okanye ekuhlaleni ixhala disorder.
Xa ezinjalo iziyobisi uphethwe "Lenuksin" (izithethantonye medicament) ibhalwa isixa mg 10 kanye ngemini. Kuncipha iimpawu zokutenxa kwenzeka ngeeveki nama-2-4. Kamva, umthamo ukuze lincitshiswe ku-5 mg ngosuku okanye landile ukuya mg-20 ngosuku.
Ngenxa lumo sisifo umbandela esinganyangekiyo, ngethuba lokuqhubeka kwekhosi unyango kufuneka ziiveki ezingama-12. Ukuthintela ukuphinda esi sifo, ingcali ukuze yabelwe kwakhona unyango, ekufuneka wenziwe zingaphelanga iinyanga ezi-6.
Hi ndlela leyi, phambi kokuqeshwa ichiza ugqirha kufuneka ingafani ukucekiswa lwentlalo kunye ukungazithembi yesiqhelo okanye ukuba neentloni.
- Ngokubanzi nexhala disorder.
Njengoko prescribers "Lenuksin" xa wabhekisela isifo? Iingcali Guest zithi ekuqaleni unyango yindlela kufuneka isetyenziswe isixa mg 10 kanye ngemini. Ukuba kuyimfuneko, idosi ukuze izazekile eliphezulu, ngamanye amazwi ukuba malunga nama-20 mg ngosuku. ukusetyenziswa ixesha elide owamkelekileyo ichiza (iinyanga ezi-6 okanye nangaphezulu).
Abantu abadala (iminyaka engaphezu 65) kufuneka lisetyenziswe kwi isiqingatha ithamo ithi ngaphantsi, oko kukuthi, 5 mg no-10 mg, ngokulandelelana (mhla).
isikhokelo ethile ngokusetyenziswa ichiza
Xa ukusilela kwezintso nganiso hlengiso idosi obubungqongo iyafuneka. Izigulana sisifo efanayo, kodwa uhlobo kakhulu, ichiza emiselweyo kubo ngobulumko obukhulu.
Xa ukukhanya okanye ukumodareyitha sisibindi Kucetyiswa idosi kwiiveki zokuqala ezimbini unyango kufuneka 5 mg ngosuku. Kuxhomekeka kwimpendulo kwalo mqulu ngomonde kweziyobisi angandiswa kabini.
Izigulana umsebenzi yehlise CYP2C19 isozyme idosi wokuqala medicament kwakhona 5 mg ngosuku. Ukuba kuyimfuneko, oko kwandiswa ku-10 mg.
Sakuba sirhoxisiwe unyango kukuba ukunciphisa ubungakanani amayeza ngokuthe ngcembe kwiiveki 1-2. Oku kuyimfuneko ukuze kuphetshwe zokurhoxa syndrome.
amacala libanda
Noko inani elikhulu labantu umbuza umbuzo wokuba nendlela ukulwa ukudandatheka ngokwabo? Ukuba iimeko ixesha elide, kodwa ayikwazi ukwenza ngaphandle abanaluncedo kwiingcali. Ngapha koko, izigulane ezifuna usetyenziso lakhula, leyo kufuneka atyumbe ugqirha.
Ukuba umntu usebenzisa yindlela wathi ukwandisa umthamo, ngoko kungekudala abe ezi mpawu zilandelayo libanda: zokudakumba yokuphefumla, iingcangcazela, unditsho, isiyezi, tachycardia, ukuphazamiseka, rhabdomyolysis, nobuthongo, lactic metabolic, isiyezi, arrhythmia, utshintsho ECG, ukugabha hypokalemia .
Kufuneka kuqatshelwe ukuba afe isiqaqa nokufa kwimeko libanda zinqabile kakhulu. Oku kwenzeka kuphela ngelixa kuphuculwa yokwamkela amalungiselelo kunye nezinye iziyobisi.
Ngenxa unyango olusetyenziswa kwiimeko libanda, unyango noncedo kwangumqondiso lavage esiswini kunye oxygenation ngokwaneleyo. Ukongeza, ukusebenza lo esweni kweenqanawa nentliziyo, kunye isixokelelwano sokuphefumla.
Drug "Lenuksin": ziziphumo ebezingalindelekanga
ziziphumo ebezingalindelekanga ekufumaneni imali bathi Idla ngokuvela ekuqaleni unyango. Emva kwexesha elithile, bona baba ayayo.
- inkqubo yokucola: ukulahlekelwa wokutya, isicaphucaphu, incasa ukuphazamiseka, ukugabha, umlomo owomileyo, urhudo, kwanda, nokuqunjelwa.
- Inkqubo luvo: nochuku, intloko ebuhlungu, ixhala, isiyezi, ukuphazamiseka, ubuthathaka, ukuphazamiseka ezibonwayo, sokulibala, ukushaya, nobuthongo, depersonalization, unditsho, iimfeketho zokufeketha, lafa, serotonin syndrome, ukuphazamiseka intshukumo, nemibono, nokubhideka.
- inkqubo Reproductive: namandla, ukuchama okungaqhelekanga, kwakunye ukunyhashwa sexesheni.
- Yesikhumba: angioedema, ebila anda, purpura, ecchymosis, pruritus kunye irhashalala,
- Jikelele: komzimba kunye nobuthathaka.
- inkqubo wokuchama: ukugcinwa womchamo.
- Heart negazi nempahla: hypotension intolerance.
- Nethe: secretion ngokwaneleyo adh.
- inkqubo Musculoskeletal: arthralgia kunye myalgia.
- uphando Laboratory: Utshintsho umsebenzi kwesibindi, electrocardiogram kunye hyponatremia.
- Komzimba: Ithuba basabele anaphylactic.
Xa imbonakalo kunye ukuqhubela phambili naziphi na iziphumo ebezingalindelekanga ngasentla kufuneka ngoko nangoko ingxelo ngayo kugqirha wakho.
Ibele nokukhulelwa
Ngaba ukusebenzisa iziyobisi "Lenuksin" ngexa lokukhulelwa? Iingcali Guest bathi, oko kucetyiswa ngenxa yokunqongophala ulwazi ngokhuseleko kunye nokusebenza kwale amayeza, sebenzisa oko ngexesha yokumitha baby. Ngaphezu koko, ukuthathwa ichiza kufuneka ayekiswe ngexesha zisanyisa.
unyango ngaxeshanye kunye namanye amachiza
izinto psychotropic, uluhlu apho kumba kakhulu, kufuneka uthathe kuphela ukuqeshwa leengcali kunye ngokungqongqo phantsi kolawulo lwayo.
Medicament "Lenuksin" nakancane ezilawulwa kunye Mao inhibitors, njengoko oku kwenza igalelo kuphuhliso serotonin syndrome. Kufuneka kuqatshelwe ukuba yokwamkela oku kuthetha abantu abatsha (ongaphantsi kweminyaka eli-24 ex-iminyaka) abagula ngengqondo kunye nokudakumba kwandisa kukuvela ideation ukuzibulala kunye sokuzibulala.
Ukusetyenziswa ngaxeshanye amayeza kunye lithium kunye tryptophan iimeko inzuzo isiphumo lokuqala ichiza
Co-ulawulo kweziyobisi kunye Hypericum perforatum kukhokelela inani elandileyo yeziphumo ebezingalindelekanga.
ukusetyenziswa ngaxeshanye i yeQela kunye anticoagulants ngqo, kunye nezinye ii-arhente ezichaphazela igazi ekunqandeni, inokuba negalelo ukuphazamiseka kwenkqubo. Kwiimeko ezinjalo, ekupheleni unyango kufuna esweni rhoqo yomguli kunye imeko igazi.
Izigulane uthathe uthe amayeza kunye arhente serotonergic, serotonin syndrome zingenzeka.
Ukudibana ne ethanol
Le medicament "Lenuksin" abufiki ethanol pharmacokinetic okanye intsebenziswano pharmacodynamic. Kodwa ke oku akuthethi ukuba yeQela zingasetyenziswa kunye notywala. Ngexesha unyango, isigulana kubhetele ukuba bashiye ukusetyenziswa kwaso nasiphi na utywala.
Kufuneka kuqatshelwe ukuba ngexesha lonyango umntu kufuneka uyeke iimoto ukuqhuba kunye nemisebenzi iintlobo umsebenzi oyingozi ukuba zifuna ukwandisa isantya lengqondo yendlela kunye ingqalelo.
Price kunye analogue beziyobisi
Kangakanani na lakhula iipilisi 'Lenuksin "? Ixabiso eli chiza inokuba nomahluko kwaye ixhomekeka eludinini. Iindleko avareji ichiza engange 990 Russian ngamnye iziqwenga 28. Uyavuma, nto kakhulu ichiza eninzi, nto leyo nayo imali bonke. Kufuneka kuqatshelwe ukuba kunqabile kuthengiswa ezikhemisti. Njengoko umthetho, emva noqeqesha ngenkqubo amayeza, ayinikiwe inikeza-odole amayeza, nto leyo uqhele kwiintsuku nje ezimbalwa.
Ngoko ke yintoni ukwenza ukuba isigulane ukuba kumiselwe i-bucala lomsebenzi, kodwa akazange abe nayiphi kwistokhwe okanye umyalelo? Kulo mzekelo, iingcali Siyaleza kuthenga elinye. "Lenuksin" aselugci- nangokomthamo kunokuba kakhulu. Qwalasela uluhlu iziyobisi enjalo ngoku:
- "Escitalopram oxalate".
- "Miratsitol".
- "Escitalopram-Teva".
- "Santsipam".
- "Escitalopram Sandoz."
- "Selectors".
- "Escitalopram".
- "Tsipraleks".
- "Elitseya".
- "Eysipi".
Ezi imali kuba oluziindleko njengoko yokuqala, kwaye sitshiphu. Noko ke, bonke zisebenza kumgaqo njengoko ichiza "Lenuksin". Ngaphezu koko, nazo ziyafumaneka kwi kagqirha. Ngoko ke, ukuthenga kubo ekhemesti ngokubona kwayo uyasilela.
Izimvo medicament
Ngoku uyazi indlela yeQela kakhulu "Lenuksin" (ixabiso). Reviews ngayo ziyabethabethana. Umntu uthi ukuba uhlangabezana njani kakuhle misebenzi, ngelixa abanye zithetha kwawo yayo.
Ukubuyekezwa Positive yale medicament eziqulathe ulwazi ukuba ngokukhawuleza nokuphelisa ixhala disorder, iphucula imo kunye nentlalo-ntle. Izigulane athi lakhula uthathe amathamo acetyiswayo uye wabavumela ukuba bahlukane lumo, ukuphakuzela uhlaselo kunye nokudakumba. Kwaye lo isiphumo nothi emva ukupheliswa ichiza.
Njengoko ngokuba ncomo ezimbi, kokukhona bahambisana kunye neziphumo ebezingalindelekanga nlichiem. Kwezinye izigulane, isicaphucaphu, ezinye intloko ebuhlungu, kwaye ezinye zange sebenzisa naliphi na ifuthe unyango.
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