Zempilo, Amalungiselelo
"Dorzopt" (wamehlo): isikhokelo, ukubuyekeza, analogs
Yiglaucoma - iqela kunokuba elikhulu izifo iliso, obubonakala ngokuba yincwadi evuliweyo ngamaxesha athile okanye esisigxina ukunyuka koxinzelelo intraocular abaneziphene zophuhliso elandelayo, yoma optic kunye ukuhla acuity olubonakalayo.
Kuba unyango lwezifo usebenzisa iziyobisi ezahlukeneyo. Amayeza iqhelekileyo "Dorzopt" (wamehlo). ncomo Consumer, imiyalelo malunga nokusetyenziswa kwale amayeza kuya kuxoxwa ngezantsi.
Ukupakisha komsindo
Kokuphi iqulethe ichiza "Dorzopt" (eye amathontsi)? Ilungu elikhutheleyo ichiza dorzolamide (njengoko hydrochloride). Kwakhona medicament iqulethe ezi izinto zilandelayo abangabancedani: Benzalkonium chloride, gietelloza, mannitol, isodiyam hayidroksayidi, citric acid monohydrate, amanzi okuhlamba.
imveliso kujongwa uveze ezineengqayi polyethylene nge-5 ml dropper umlomo.
pharmacodynamics
Yintoni wamehlo "Dorzopt"? Guide ingxelo ukuba esi sixhobo i anhydrase గుర్తులు ibhaloni lendawo inhibitor. Kuye nefuthe ngxelo imbi kwi secretion intraocular cerebrospinal kunye abangaphangeliyo ukuyilwa hydrogen carbonate kunye namanzi buthathaka ukudluliselwa kunye sodium.
Eli chiza akubangi miosis okanye ukungaboni ebusuku, kwakunye spasm yokuhlala.
Pharmacokinetics
ingaba ichiza ako, "Dorzopt" (wamehlo)? Kukufakwa ichiza kwenzeka ngokusebenzisa inwebu ngokusebenzisa kwesebe kunye sclera. rates ukufakwa systemic echiza iphantsi kakhulu.
Ngenye egazini, eyona nto esebenzayo ichiza ungena ngokukhawuleza kwi iiseli ezibomvu ezinomthamo eliphezulu anhydrase గుర్తులు ibhaloni 2.
Unxibelelwano kunye iiproteni plasma kwenzeka ngo-33%. Ichiza atshintshelwe N-dezetilirovanny metabolite, nto leyo esebenza kakhulu anhydrase గుర్తులు ibhaloni 2, kodwa iyakwazi kuthintele anhydrase enye గుర్తులు ibhaloni.
ukusetyenziswa elide ichiza kukhokelela nokwanda yayo erythrocytes.
Wabonisa amayeza nge nezintso. ukususwa kwawo 2 ukupheliswa Inqanaba: fast and kade. Le yokugqibela ebangelwe ukukhululwa chu lecandelo esebenzayo iiseli ezibomvu zegazi.
nesiqingatha sexesha-ubomi iinyanga 4.
ubungqina
Xa prescribers "Dorzopt"? wamehlo ziyasebenza kakhulu unyango ephakamileyo uxinzelelo intraocular xa abantu lwegazi ocular okanye neglaucoma evulekileyo-pseudoexfoliative (kuquka eziziisekondari).
Izimo
Ziziphi iimeko, awukwazi ukusebenzisa iziyobisi "Dorzopt"? wamehlo ukuba ungamiselwanga ukuba:
- lactic hyperchloraemic;
- Hypersensitivity ukuba izinto abasemthethweni;
- ukuphazamiseka kidney kakhulu;
- njengomntu;
- kwithuba zisanyisa.
Ngononophelo kakhulu kufuneka kusetyenziswe le sixhobo:
- diabetes;
- izigulane ongaboniyo hepatic;
- abo ingxinano encinane iiseli inwebu endothelium lwalo (of amathuba aphezulu nokudumba kwenwebu yamehlo).
umthamo
Yabela isixhobo eyaziswa ukuba unyango lwezifo neso oyingcaphephe elimxinwa kuphela emva kokuba kugqitywe uviwo ngenyameko isigulane. Gqiba ekuqulunqeni desirably enye ukuhla ukuya kwi sac conjunctival ka kathathu ngemini.
Ngenxa ukuhlanganiswa iziyobisi kunye beta-blocker kweziyobisi mlonyeni ukusebenzisa enye idrophu kabini yonke imihla.
Ukuba unyango lwezifo ocular luquka izinto eziliqela lwamehlo, lekhefu phakathi instillation yabo kufuneka imizuzu ubuncinane elishumi.
imiphumela emibi
Ukuba usebenzisa wamehlo "Dorzopt" Ukusabela beenqila balandelayo ukuze aphuhlise kwizigulane:
- Ukurhawuzelelwa, baqhumisela imvakalelo emehlweni, conjunctivitis, paresthesia, nokudumba ijwabu, kujuba blepharitis, ukucaca kakuhle yombono, photophobia ezingekhoyo punctate keratitis.
- kunqabile kakhulu isicelo beziyobisi zezi: iridocyclitis, ukwandisa ububanzi inwebu, nokwaliwa, hypotension iliso kunye ngamava semehlo emva antiglaukomatoznyh imisebenzi.
ziphumo bezingalindelekanga zeNkqubo:
- imvakalelo isicaphucaphu, incasa ekrakra emlonyeni, uphuhliso nefrourolitiaza, ukudinwa, migraine, amabi, exudative erythema multiforme, ityhefu epidermal necrolysis, igazi aplastic, irhashalala ulusu kunye agranulocytosis.
amacala libanda
Ziziphi iimpawu kwenzeka xa usebenzisa "Dorzopt" ngeedosi eziphezulu na ichiza? Eyedrops, analogs leyo ziboniswa ngezantsi, nesandla:
- lactic uphuhliso;
- ukuphazamiseka kwamanzi kunye nemali electrolyte;
- CNS imiphumela emibi.
Kuba unyango ezinjalo iimeko abaqeshwe symptomatically, sikhatshwe kolawulo umgangatho electrolytes kunye pH negazi.
imithi
- Xa kudityaniswe arhente antiglaucoma ichiza (beta-blocker, "dipivefrin", "pilocarpine", "Carbachol") inyusa ukusebenza kwayo.
- With "acetazolamide" kwandisa amathuba yeziphumo ebezingalindelekanga lwenkqubo.
- Kunye iidosi ezinkulu acetylsalicylic acid kwandisa ubuthi ichiza.
izincomo ezithile
Ukusetyenziswa iingqayi multidose ukukhala uphuhliso keratitis yebhaktiriya. Oku kungenxa kungcoliseko ngabom kwiziqulatho zazo.
Ngexesha unyango "Dorzoptom" kufuneka asebenzise iilensi benzalkonium chloride kunokuba ziyityhefu kwaye kubangele ubuhlungu emehlweni.
Analogs kunye nexabiso neziyobisi
Buyisela ichiza uthathwa iliso kungenziwa ngeendlela ezifana 'Trusopt "yaye" Floksal ". Price of ichiza malunga 350 engange.
ukubuyekeza yabathengi
Ngelishwa, ukubuyekeza kwabathengi malunga ichiza "Dorzopt" zinqabile. Phakathi okulungileyo kule inqaku iziyobisi ezifana nobukho kunye nokusebenza. Noko ke, abanye abathengi reactions ochaphazelekayo, basekuhlaleni systemic ezingalunganga ukuba zenzeke ngexesha unyango kunye ngamathontsi. Kule nkalo, iingcali ukuncoma ukusetyenziswa kweziyobisi phantsi kwegama "Dorzopt Plus".
Eyedrops zikhankanywe ngasentla ziquka into ezongezelelweyo ezifana, ezifana timolol. Ixhasa kutsalwe ulwelo intraocular.
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