ZempiloAmalungiselelo

"Amlodipine": yintoni esiza, imiyalelo ukusetyenziswa, analogs, ncomo

Yintoni lwegazi? Impendulo yalo mbuzo yaziwa kubantu abaninzi, ingakumbi abantu abadala. Njengoko usazi, oku ukunyuka ziqhubeke uxinzelelo lwegazi, apho izalathisi baphawula ezifana 150/90 mmHg. Art. nangaphezulu.

Kukholelwa ukuba lwegazi yeyona sifo kakhulu kwinkqubo sentliziyo. ukwanda ziqhubeke uxinzelelo lwegazi uyaqapheleka 25-30% yabantu abadala. Hi ndlela leyi, iminyaka sisifo ndiyibonile 55-65% yabantu.

Kutheni kukho lwegazi? Le nto inokwenzeka ngenxa yezizathu ezininzi. Ngokufuthi abadala xi liphuma ngenxa yobunzima ngokwasengqondweni iimvakalelo. Ngako oko abantu ezithandwa lwegazi, kufuneka kube ukuzola.

Asikwazi ukuba esi sifo kaninzi kwenzeka ngenxa yokuba umzimba, ubudala, isini (common kakhulu kwisiqingatha wamhle lobuntu), ngokugqithiseleyo ukutya ityuwa, ukutya gipokaltsievoy, ukusebenzisa kakubi utywala, imfuza, ukutyeba, ukutshaya, isifo seswekile kunye t. d.

Ingaba kuyimfuneko ukunyanga wegazi? Oogqirha bathi xa uziva mnandi, izigulane kufuneka uqinisekise ukuthatha amachiza kuthoba uxinzelelo lwegazi. Kuba omnye wabo ukuthwala neziyobisi "Amlodipine". iziphumo ebezingalindelekanga kwesi sixhobo, iimpawu zayo, ixabiso, kunye analogs zidweliswe ngezantsi.

Inkcazelo ngemveliso amayeza, ukwakhiwa kwayo nokupaka

Ziziphi fomu yenziwa iziyobisi "Amlodipine", ixabiso apho zidweliswe apha ngezantsi? Ingqalelo ichiza eveliswa ngokohlobo amacwecwe ifomu emhlophe kunye ploskotsilindricheskoy. element kwakhe yangoku amlodipine.

Le ekuqulunqeni kuthengiswa esiseleni nentaba (tablets 10) apho zipakishwe kwiibhokisana.

Indlela yesenzo iziyobisi

Ntoni na "Amlodipine"? Ngokutsho imiyalelo, ichiza liveza iipropati iqapheleka umfutho kunye antianginal. Ngaphezu koko, akukho nto ukunika nabo calcium ndzulu inwebu iiseli engabalulekanga kunye neeseli nemithambo.

Yintoni na ichiza "Amlodipine"? Ukususela oko kunceda eli yeza? Kuhle kunciphisa uxinzelelo oluphezulu lwegazi. Oku kungenxa yokuba ubuchule ichiza lokwandisa imithambo yegazi.

Kufuneka kuqatshelwe ukuba ingqalelo ichiza ebonisa isiphumo antianginal. Le impahla ichiza ibonelelwa element yayo yangoku. Oogqirha ingxelo ukuba amlodipine enkulu kuphela arterioles (peripheral), kodwa kwakhona kunciphisa ukuxhathisa peripheral nemithambo. Lapho wathi nto ayithethi ukuba tachycardia (reflex).

Yintoni umphumo ngokusebenzisa ichiza "Amlodipine"? Yintoni eyenza le sixhobo? Ngenxa eli chiza intliziyo yomntu iqalisa osebenzisa amandla eninzi kwaye kakhulu kunciphisa imfuno ioksijini engabalulekanga.

Kinetics kabi

Drug "Amlodipine" uxinzelelo (ophezulu) ifunxwe ukusuka emathunjini ngokucothayo kakhulu, kodwa ngokupheleleyo. Le Incopho abasuka zithako yalo egazini kuphunyelelwa emva kweeyure 8.5. medicament Plasma protein esibophelelayo nama-98%.

Le medicament "Amlodipine", apho inyathelo sibhekiswe zokucutha, ivavanywa ukutya ezincinci. Kule fomu yezabelo leyo abe umsebenzi imithi ephantsi. Umzimba neziyobisi xa edlula esibindini.

I-avareji isiqingatha-ubomi amlodipine kunye nezakhi zawo iiyure eziyi-36. Xa kuphakanyiswe ngamandla uxinzelelo ngegazi ixesha kwandiswa ukuya kwiintsuku ezimbini, abadala - ukuya kutsho kwiiyure ezingama-66, yaye zesibindi nokuphazamiseka - ukuya kutsho kwiiyure 58.

Lithathwe kweziyobisi ngohlobo metabolites ngokusebenzisa amathumbu kunye nezintso.

Drug "Amlodipine": yintoni esiza?

Kwezinye iimeko, iyeza zisenokuthathwa ukuba eyabelwe isigulane? Izinto ezibonisa ukuba yokwamkela imali lithi zilandelayo:

  • angina ezinzile;
  • vasoconstriction okanye vasospasm;
  • angina vasospastic;
  • Umfutho wegazi (njengoko monotherapy okanye zidityaniswe namanye amachiza);
  • cardiomyopathy nonischemic inimba.

Kwezinye iimeko, ichiza iye "Amlodipine" kungenziwa recommended? Yintoni eyenza eli chiza? Idla emiselweyo kunye namachiza antianginal, kuquka izigulane abanganyangekiyo unyango ibeta-blocker okanye nitrate.

Siphelisa yokwamkela ichiza

Ngoku uyazi injongo apho izigulane kufuneka ufumane i "Amlodipine" iipilisi. Ezibonisa eli yeza edweliswe apha ngasentla.

Ngokuphathelele Izimo, ukusetyenziswa kweli chiza akuvumelekanga ukuba hypotension. Ukongeza, oko singacebisi ukusetyenziswa umntwana, kwakunye phambi hypersensitivity izithako yayo.

Kufuneke njani amayeza "Amlodipine"?

Analogue, ixabiso eli chiza zidweliswe ngezantsi.

Indlela lwezifundo apha lolawulo ngomlomo. Le umthamo ichiza ibalwa ugqirha, ngokuxhomekeke imeko yesigulane.

Izigulana lwegazi (lwemithambo) kunye nedosi angina Minimal beziyobisi ngosuku 5 mg. Ukuba kuyimfuneko, kwi kulandelayo kuyenzeka ukuba anyuse imali ngqo amaxesha ezimbini, oko kukuthi, ukuba bayinyuse ku-10 mg ngosuku.

Xa unyango lwe cardiomyopathy inimba medicament esebenzayo Kucetyiswa ukuba athathe idosi ye 2.5 mg. Ukuba amayeza kakuhle wabunyamezela isixa angandiswa izihlandlo ezine.

Ngokutsho iingcali, zidlule iidosi abawacebisayo ichiza (ngaphezu kwama-10 mg ngosuku) akukhuthazwa ekubeni oku kunokukhokelela iziphumo ezingafunekiyo.

Reception "amlodipine" kubanjiswene ne beta-blocker, womchamo (thiazide) kunye ACE inhibitors ayifuni uhlengahlengiso balawule.

Iintshukumo ngu-lomsebenzi

Njengoko sihambisane "Amlodipine 'iziyobisi? ziziphumo ebezingalindelekanga ezivela kweli chiza azinako bengekho. Noko ke, kwezinye iimeko (umzekelo, ukungathobeli idosi), oko zisabangela:

  • tachycardia, hyperplasia gingival, yokucoca, ukozela;
  • arrhythmia, isicaphucaphu, iyangongoza, intloko ebuhlungu, ukuphelelwa ngumphefumlo;
  • intlungu ezibukhali esiswini, nokudumba peripheral, nokudinwa;
  • hypotension, irhashalala, paresthesia, pruritus, ukuba nesiyezi.

Kufuneka kuqatshelwe ukuba ulawulo ezigulo ezondeleyo ingqalelo tablets, isiguli iintlungu kwi imilenze.

Amacala libanda, iziyobisi

Ulwazi malunga amayeza amatyala libanda, idatha ayifumaneki namhlanje. Nangona oonoklinikhi lubonisa ukuba xa efumene isixa esikhulu beziyobisi izigulane ukubonisa ngayo kwicala elide.

imithi

Ngaba kuvumelekile ukuba kunye namanye amayeza ukuba uthathe amayeza "Amlodipine"? Imiyalelo, izimvo kwiingcaphephe athi isiphumo iqinile beziyobisi ngakumbi xa zidityaniswe kunye blocker calcium channel. A ofanayo kulindeleke ngokusebenzisa indlela ilungiselelwe inhalation zomzimba, kunye orlistat. Phela, indibanisela enjalo nokuba bamqumbise enengxaki unesifo.

Okwehlileyo antigipetrenzivnogo ukusebenza nokugcinwa sodium emzimbeni womntu kuvandlakanywa kunye neepilisi "Amlodimpin" estrogen kunye sympathomimetics.

Uphuhliso iimpawu ezinjalo neurotoxicity, njengoko ukuduma, isicaphucaphu, Ataxia, ukugabha kunye norhudo, zibangelwa yi ulwamkelo ngaxeshanye amlodipine kunye Lithium carbonate.

usebenzisa amayeza kwaye kwaqwalaselwa "Indomethacin", kunye nezinye NSAIDs kunciphisa isiphumo umfutho lokuqala.

Ibele nokukhulelwa

Ukhuseleko lwamayeza "Amlodipine" ngexesha lokukhulelwa awuthunyelwanga efunda. Kukwasebenza kwanjalo kuyo ithuba zisanyisa. Kulo mba, imveliso wathi kwiindawo ezinjalo kufuneka zisetyenziswe kuphela xa ubungozi obunokubakho umntwana ngaphantsi kakhulu luncedo impilo kamama.

iingcebiso Jikelele ulwamkelo ichiza

IMimiselo olubekwe emacwecweni, uthi kufuneka athathwe ngononophelo kakhulu waphula umthetho kwesibindi kunye nezintso, kwakunye stenosis aortic.

Ukulungiswa ithamo ukuba sele kuchaziwe ngentla, abadala abayi efunekayo.

Le medicament "Amlodipine" zingasetyenziswa kunyango kwizigulane kunye une cardiomyopathy inimba (nonischemic), nto leyo sikhatshwa ukusilela intliziyo (uhlobo ezingapheliyo).

Izifundo lwezonyango ngokusetyenziswa eli chiza xa izigulane ezingabantwana azikhange kuqhutywa.

Imiqathango yentengiso kunye nokugcinwa, ukuba kuthengiswa

Ukugcina olu nyango kufuneka ibe kwindawo, kwindawo emnyama eyomileyo apho lobushushu awudluli degrees 25, kwaye apho kungekho ukufikelela kubantwana abancinane.

Lipapashwe kulo ndawo ngaphandle kagqirha kagqirha. Ngokutsho umyalelo, ubomi ezikhabhathini ziinyanga ezili-24. ukuthatha iyeza emva kokuphela kwale xesha akuvumelekanga.

Iindleko amayeza ezikhemisti kunye amalungiselelo ezifanayo

Kangakanani na 'Amlodipine "icwecwe? Ixabiso le mveliso zinokuba nomahluko, kodwa kunjalo akukho phezulu kakhulu. Namayeza umthamo we-10 mg ixabisa malunga ne-55 engange, kwaye umthamo we-5 mg - malunga 35 engange.

Njengoko kukhankanyiwe ngasentla, hypertension sisifo eqhelekileyo kakhulu. Ngoko ke, iinkampani ezixuba amayeza ukuvelisa iziyobisi minyaka yonke ngakumbi nangakumbi yenzelwe ukuthoba uxinzelelo oluphezulu lwegazi. Hi ndlela leyi, elikhethekileyo nezixhobo zokunika ingxelo, zininzi. Oogqirha bathi iipropati umfutho ezi uphawu lwamayeza zilandelayo: "Agen", "Tenoks", "Akridipin", "Stamlo M", "adipic", "Stamlo", "Amlo", "normodipin" "Amlodipine Sandoz", " Omelar Cardio "," Vero Amlodipine, "" Norvasc "" Amlodipine-Teva "," Cordy Kor "," Amlodak "," Norvadin "," Amlovas "," Korvadil "," Amlodigamma "," cardilopin "," amlodipine Alkaloid "," Karmagip "," Amlodhi "," Kalchek "" amlodipine Zentiva "," Amlonorm "" amlodipine-Agio "," Amlotop "" amlodipine Cardio "," Amlorus "," Amlodifarm "" amlodipine besylate "," Amlong "," Ngaba lokard-Sanovel "kunye t. d.

Izithuba iziguli noogqirha

Nge ubudala, izifo ezifana lwegazi, ufakwa elandayo inani labantu. Njengokuba sisazi, le meko luphawulwa mpawu zilandelayo: nesiyezi, ukudinwa ngokugqithiseleyo, intloko ebuhlungu, ukutyhafa, mnyama amehlo, ukozela, kwaye ngaphezulu. Ngokutsho kweengcali, zonke ezi mpawu zinyamalale kwisithuba iiyure ezimbalwa emva kokutya "Amlodipine" amacwecwe ithamo mg-5 okanye 10.

Oogqirha ingxelo ukuba ichiza ekuthethwa yenye ndlela ikhawuleza nolusebenzayo. Xa ixesha elifutshane bexesha omeleza uxinzelelo lwegazi yomguli, kwaye iphucula kakhulu imeko yayo jikelele.

Ke kubathengi, bathi ke indlela elula isicelo nokumila esi sixhobo phakathi iimpawu. Ukunciphisa uxinzelelo oluphezulu lwegazi, kufuneka isigulane ukuba athathe ipilisi enye. Ngoko ke amagqirha zilumkisa ukuba le libanda chiza inokuba negalelo okanye ukuphucula ukubonakala basabele ezibi. Kulo mba, azikho kucetyiswa ukuba asebenzise ngaphezulu kwe-10 mg beziyobisi ngosuku.

Kufuneka kwakhona uqaphele ukuba inani elikhulu labathengi abonwabileyo ixabiso eliphantsi yathi kuthi, njengokuba kwakunye nokufumaneka kwayo kuzo zonke ezikhemesti ukukwazi endaweni oothixo.

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