Zempilo, Ukulungiselela
Iidakamizwa "I-Scopolamine hydrobromide": iipropati, izibonakaliso kunye nokuchaswa kokusetyenziswa
"I-Scopolamine hydrobromide" yileyeza esetyenziswa kakhulu kwiyeza zanamhlanje. Kodwa, ke, izigulane zinomdla ngolwazi olongezelelweyo, ngokukodwa, iipropati zezilwanyana, izibonakaliso kunye nokuchasene nokunyango, njl njl.
Isilwanyana "I-Scopolamine hydrobromide": umyalelo, ukubunjwa kunye nefomu yokukhululwa
Ukuqala oko kuyimfuneko ukuqonda ukubunjwa kweyeza. "I-Scopolamine hydrobromide" (iresiphi yesiLatini - iScopolaminum Hydrobromicum) i-crystals ebalabala. Enyanisweni, iyakuthi ibonakale ngesimo se powstalline powder kunye nesimo esichukumisayo emva kokuhamba. Ixabiso lenzeke ngokukhawuleza kwi-alcohol kunye namanzi. Ngendlela, eli qela lilo liqela le-alkaloids - itholakala kwizityalo ezifanayo njenge-atropine - i-bleached, scopolia, belladonna, udope.
Kwimveliso yekhemist ingathengwa kwifom powder. Kodwa ngokuphindaphindiweyo isilwanyana sisetyenziselwa isisombululo se-0.05% - ithengiswa kwii-ampoules zeglasi ezili-1 ml. Kukho iibhotile ezi-5 okanye i-10 ml - esi sixa sine-methyl cellulose. Ampoules (okanye izitya) kufuneka zigcinwe kwindawo epholileyo, apho ilanga elithe ngqo lingafi. Ubomi beShelf - iminyaka emi-5 ukususela kumhla wokuveliswa.
Inkqubo yesenzo sonyango
I-Scopolamine hydrobromide ine-effect effect efana ne-atropine-isebenza ngokumalunga neenkqubo ze-cholinergic. Ngokomzekelo, isigulane emva kokuba sithathe iyeza elithe lakhubazeka ngethuba lokuhlala, ukunyuka kwentliziyo, ukunciphisa ukufihla, kunye nabafundi abahlanjululwayo kunye nokuphumla kwezihlunu.
Kodwa kwinkqubo yesantya ephakathi, iyakwenza ngokuhlukileyo, enye inqanda umsebenzi wayo. I-Scopolamine inqanda ukuhanjiswa kweempembelelo zesigulane esivela kwipatramidal tract ukuya kwizakhiwo zomqhubi kwintambo yomgogodla. Ukongeza, i-arhente ivimba i-cholinoreactive receptors kwisakhiwo esicacileyo. Yingakho isilwanyana sinomdla (sedatives) kunye nomphumela wempembelelo emzimbeni womntu - kunciphisa umenzi wemoto. Ngendlela, enye yezinto ezi zinto zilandelayo kukuba emva kokuthatha, njengomthetho, kukho i-short-term amnesia - umntu akhumbuli oko kwenzekayo.
Kwiimeko ziphi izilwanyana ezisetyenziswayo? Iinkcazo
Eli seziyobisi lisetyenziselwa kwamagatsha amachiza amaninzi:
- Njengoko isisombululo sokukhusela kunye nesalathisi sokusebenzisa i-anesthetic isisitoreji sisetyenziselwa ukuqhutyelwa komzimba kunye nokuhlinzwa ukuze silungiselele i-anesthesia.
- Kwiingxaki ze-neurology zokuthatha izidakamizwa zi-postencephalitic parkinsonism kunye nokuthuthumela ukukhubazeka.
- I-Ophthalmologists nayo isebenzisa le nkunkuma ngendlela yamaconsi ehlohlo - iyasebenza kwi iridocyclites kunye ne-irites. Amaconsi asetyenziswayo xa kukho isidingo sokwandisa umfundi wegulane (umzekelo, ngaphambi kokuba kulandelwe iinkqubo).
- Iyeza lifumene isicelo saloo-psychiatry, kuba lisebenza njengesilwanyana.
- Xa kwenzeka ukugula komoya kunye nolwandle, "i-Scopolamine hydrobromide" inceda ukujamelana nokukhwabanisa, ukuhlanza nokukhathazeka. Le khemikhali isetyenziswe kwisibisi "i-Aeron".
Ukusetyenziswa kwe "scopolamine hydrobromide" kunceda ukujamelana neengxaki ezininzi. Nangona kunjalo, unokwenziwa kuphela ngudokotela oya kwi-adnesis emva kokuba enze i-anamnesis kwaye afumane yonke idatha yokuxilonga.
Isiyobisi "Scopolamine hydrobromide": imiyalelo yokusetyenziswa
Njengoko sele kuthethwe ngaye, isilwanyana sikhululwe njengesisombululo - injected okanye phantsi kwesikhumba okanye nge-intramuscularly. Umthamo wezonyango weziyobisi (xa kuziwa kwi-injection subcutaneous) ukusuka ku-0.0002 ukuya ku-0.0005 g scopolamine. Ngokuqhelekileyo, izigulane zinikezwa i-0.5 okanye 1 ml yesisombululo se-0.05% - iilenki zenziwa ezimbini okanye kathathu ngosuku.
Ukuba sithetha ngamaconsi asehlohlo, izigulane zibekwe phambi kwe-1-2 kwizame nganye. Inkqubo kufuneka iphindwe kabili ngosuku, isebenzisa isisombululo se-0.25%. Kubalulekile ukuqonda ukuba eli lonyango elinamandla kunye nokungagunyaziswanga kwalo, isicelo esingenakunceda singakhokelela kwiingxaki eziyingozi kakhulu. Ugqirha kuphela onokumisela isilwanyana, umisele isigqirha, umisele umyinge kunye nobude bekhosi.
Ngaba kukho naziphi na izithintelo kunye nokuchasene?
Ingaba kuyimfuneko ukuyimisela kuzo zonke iindidi zabantu umkhiqizo weyeza "Scopolamine hydrobromide"? Enyanisweni, iziyobisi zinemiqobo. Ayikwazi ukulawulwa zizigulane ezinezifo eziphilayo zesimo senhliziyo.
Kuluhlu lwee-contraindications lubandakanya isifo sikashukela kunye ne-glaucoma. Ungasebenzisi iyeza ukuze uphathe izigulane ezinezifo ze-thyroid, ngakumbi i-hyperthyroidism. Amadoda ane-hypertrophy yeprostate esi sixombululo sinokulimaza. Isicelo esele sikhulile, kodwa silumke kakhulu ukwenza oku.
Iziphumo ezinokubakho zonyango
Ngokutsho kwedatha yeenkcukacha, le michiza kwiimeko ezininzi iyakunyamezela. Nangona kunjalo, ezinye izigulane zihlakulela umphumo. Ngokomzekelo, kukho ukuphazamiseka kwindawo yokuhlala kwilensi kunye nokuphucula okuqhubekayo kwabafundi, okuchaphazela uvakalelo ekukhanyeni nasekuboneni izinto ezibonakalayo.
Ezinye izigulane zikhalaza nge-tachycardia, i-palpitation palpitation. Ukuphendula kwangasese kubandakanya ukungcola, umlomo owomileyo kunye neengxaki zokucoca. Ngamanye amaxesha, xa umthamo ukhethwe ngokuchanekileyo, unyango lusebenza ngokugqithiseleyo - umntu uyaba neentloni, ukukhohliswa kunye neengcamango zivela. Ngokuqinisekileyo, xa kwenzeka ukuphazamiseka okuchazwe ngasentla kubalulekile ukujongana nodokotela oya kubakho njengentuthuko yeengxaki ezinokwenzeka.
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