Zempilo, Amalungiselelo
Ichiza "Antistius": analogue, imiyalelo esetyenziswa kunye nengxelo
"Antistius" (international igama non-wezindlu - trimetazidine) - uye Antihypoxanth inyathelo. Ephelisa hypoxia nge nokubuyiselwa yokucolwa amandla abaqhelekileyo kwi iiseli, umqulu ukulingana phakathi ioksijini engenayo kunye othe waphuma. IZenzo phezu luvo kunye cardiomyocytes ingqondo, banikwe izinto eziyimfuneko.
Iibhloko landa secretion ye asidi ezinamanqatha, ezo ezibangela ezinkulu iingxaki ukutya yeselula. Heart kwemisipha buyasikhulula, ngaloo ndlela inegalelo nokuzinziswa kwamathumbu engabalulekanga. It kwandisa imifinya iseli, nokuthintela nokwanda kuwo of ion potassium, calcium sodium.
Pharmacokinetics
Le into esebenzayo (trimetazidine) ngokukhawuleza kwaye phantse ngokupheleleyo wendele inani kwinkqubo yokwetyisa. Digestibility "Antistius" phantse 90%. Ukuphumeza umxholo ubuninzi egazini yenziwa iiyure ezi-2. Lula uleyisayo imiqobo phakathi kwegazi kunye namalaphu. Ukubambana kwiiproteni plasma yi-16%. Kwazona ngokusebenzisa izintso (60% - in isimo sokuqala). ngokupheleleyo ixesha ukuphelisa imalunga ne-14 iiyure. Abantu abadala ngaphezu kweminyaka eyi-65 ezithatha ichiza, liyatshona ixesha ukuzala ukuya kwiiyure ezingama-24.
ifomu Release komsindo
Ukulungiselela "Antistius CF" 35 mg № 60 (analogue ingafunyanwa kwi idosi enye) ekuveliseni ngokohlobo biconvex, amacwecwe ngeenxa zonke. Nguwuphi zipakishwe phezu izikhongozeli ezikhethekileyo polymeric. "Antistius" tablet nganye iqulathe lamanqanaba ezimbini: i ngumongo ngaphakathi okanye nombala omhlophe okanye tyheli, iqokobhe ngaphandle iye unelupus. Kwenye tablet "Antistius" eziqulathwe 20 mg ukwimo esisiseko - trimetazidine dihydrochloride.
Ukubunjwa kwakhona iquka amacandelo abancedisayo, apho zimelwe wemagniziyam stearate, hypromellose, triacetin, intsimbi oxide ebomvu naziiperile, ngenxa microcrystalline kwincindi.
Imiyalelo "Antistius"
Ukukhonza ngaphakathi kwi umthamo we 40-60 mg, yahlulwe 2-3 nasebusuku. Ngokuxhomekeka kuhlobo kunye nobungozi besi sifo kwimeko nganye amisele ikhondo ekhethekileyo unyango.
isicelo
"Antistius" isetyenziswa:
- unyango lwexesha elide ischemia kwentliziyo: isilumkiso yokuhlaselwa angina kunokwenzeka (njengoko ichiza okanye nayiphi na izithako nothomalaliso zidityaniswe ezimeleyo).
- Therapy umonakalo inkqubo vestibular kunye organ ukuva (in t. H. Vertigo, ukuduma, bakuva umonakalo).
- izilonda nemithambo umbono.
imiphumela emibi
A lot of izigulane osebenzisa isiyobisi, kukho ukunyamezelana eliphezulu.
Ayifane yenzeke, kodwa kukho ezinye iziphumo ezingafunekiyo:
- phezu inxalenye iphecana zesisu - ukuphazamiseka sotyatyazo, iintlungu esiswini, isicaphucaphu, ukugabha, ukuphazamiseka sorhudo;
- umonakalo luvo inkqubo, cranialgia abonisa, iintshukumo discoordination ukusilela iimpawu extrapyramidal abakreqayo ukusilela ukusuka 'Antistius ";
- yenhliziyo - ukuthoba uxinzelelo, iyangongoza, kukuvela arrhythmias;
- kunciphise inani zegazi kwenzeka agranulocytosis;
- kunokubangela iziphumo dermatological ngohlobo irhashalala komzimba kunye ukurhawuzelela kolusu.
Kwiimeko ezinqabe kakhulu, a hepatitis ityhefu.
Besebenzisa "Antistius" azivumelekanga:
- abasetyhini abakhulelweyo;
- ngexesha lokuncancisa;
- abantwana abafikisayo;
- ne umsebenzi othile sezintso;
- xa kwimeko hypersensitivity nobandlululo kwezinye iinxalenye ngamnye yokulungiselela.
Sebenzisa ekhulelwe kwaye ngexesha lokuncancisa
Iimvavanyo izilwanyana lubonise ukuba "Antistius 'inokuba neziphumo eteratogenic ekukhuleni kosana olungekazalwa. Noko ke, ngenxa yokuba imali eyoneleyo ulwazi malunga ilunyango olukhuselekileyo "Antistenom" ngexa lokukhulelwa, amathuba kukuvela ukungaqheleki ezahlukeneyo kuphuhliso ezingekazalwa ayikwazi ngokupheleleyo kwaba njalo. nto abafazi abakhulelweyo ekuqeshweni iyeza ayisetyenziswanga unyango.
Kwakhona engazimisele nokuba "Antistius" ibe ubisi lwebele. Ukuba isiqu "Antistius" kuyimfuneko, kuyimfuneko ukuba uyeke ukuluncancisa.
Ayivunyelwanga ukusetyenziswa ebantwaneni.
Intsebenziswano kunye namanye amachiza
Not wafumana imiphumela intsebenziswano "Antistius", kunye nokuqeshwa yayo ngaxeshanye kunye namanye amayeza.
Okwangoku, oko akubonisi ityala olunye libanda, iziyobisi "Antistius" yemiyalezo. Analogue beziyobisi isetyenziswa ngokubanzi.
oyi
"Antistius" 35 mg (kubandakanywa analogs) elawulwa ukwenzela ukuthintela uhlaselo angina kunokwenzeka, kodwa ayikwazi kusetyenziselwa isiqabu. Akucetyiswa ukuqeshwa "Antistius" ngenxa isanda kwi ukunyanga isifo sentliziyo okanye angina ezingazinzanga.
Akuvunyelwanga ukusetyenziswa ngaxeshanye kotywala kunye nonyango "Antistenom" kuba izithako ezisebenzayo na uhlobo malunga zempembelelo (ethanol kunye trimetazidine). Ukuba uluphosile iindlela enye okanye ngaphezulu amayeza, akavumelekanga ukuba bayisebenzise ngeedosi eziphezulu isicelo elandelayo.
"Antistius" alunasiphumo kwi izinga yokusabela yaye oko kubangela ukozela, ngoko ingasetyenziswa kulawulo endleleni.
Impilo "Antistius" ziinyanga ezili-36 ukususela kumhla wokwenziwa. Sikugcine ezomileyo, epholileyo ingafumaneki abantwana. Ekhuselweyo elangeni. Ayikwazi kusetyenziswa emva komhla wokuphelelwa, njengoko kusenokuba ziyakwehlisa ngokubonakalayo impumelelo okanye enze iimpawu ezingafunekiyo.
Yintoni indawo ichiza?
On efumanekileyo kwi "Antistius" kunoogxa iziyobisi. Izimvo kuzo esihle kakhulu. Mhlawumbi ukusetyenziswa kweziyobisi, efana "Antistenom" indlela action:
- iintyatyambo hawthorn;
- "Vazomaga";
- "Histochrome";
- "Dinatona";
- "Dibikora";
- "Doppelgerts Kardiovitala";
- "Ezafosfina lyophilisate";
- "Idrinola";
- amalungiselelo camphor;
- "Kardionata";
- "Qudesan";
- "Mexicor";
- "Meldonium";
- "Mildronate";
- sodium adenosine triphosphate;
- Neoton lyophilisate;
- "Orokamaga";
- "Riboksin";
- "Serotonin";
- "Taufon";
- "Ubinone";
- "Firazira" okanye "Fosfadena".
"Antistius": nabalingani Russian
- "Angiozyme kunamandla." Kuyinto kakhulu efikelelekayo, kodwa kanye njengokuba Ndisomelele "Antistius" (nucleoside cheap zingathengwa na ekhemesti). It obunamanani enkulu yeziphumo ebezingalindelekanga.
- "Vero trimetazidine" - siyobisi enganeno.
- "Deprenorm MV" - ngokuqesha kwakhe kwenzeka effects ngakumbi, kuyabiza.
- "Medarum" - phantse akukho ziziphumo ebezingalindelekanga, kodwa ichiza ibiza kakhulu kwamanye amaxesha.
- "Rimekor" - kukho ixesha elide amanyathelo, aqhelelkileyo yeziphumo ebezingalindelekanga, enganeno.
- "Karditrim" - i ziphumo bezingalindelekanga eqhelekileyo ngakumbi, kunoogxa imali eninzi.
- "Tridukard" yaye "Trimektal" engasebenzi kakuhle, nto ke leyo ebangele ukuba kufuneka ingasetyenziswa xa abantu bokubabambela, ichiza "Antistius".
Analogs nawethutyana, amazwe
- "Metagard" - xa kutyunjwa rhoqo uneziphumo ebezingalindelekanga, yinto analogu ebizayo
- "Predizin" - iziphumo ezingalindelekanga rhoqo.
- "Trimetazid" - lineziphumo ebezingalindelekanga ezimbalwa.
- "Prekard" - uguqulelo cheap kodwa ngaphantsi olusebenzayo.
- "Trimetazidine-Teva" - ichiza olubiza kakhulu.
reviews
"Antistius" (njengoko analogue) rhoqo ezisetyenziswa kunyango mihla, ngenxa yoko, ingxelo elingafaniyo kakhulu. Uninzi lwezigulane uthetha "Antistene" njengendlela indlela ephumelelayo kakhulu.
Iyeza incede izigulane ezininzi ingxelo ukuba imeko yabo jikelele yaphucuka, ukulala yaphila, uxinzelelo lubuyele kwisiqhelo. Ukwandisa amandla ubomi. Ichiza Ususa vertigo kunye ingxolo entloko. nokuphazamiseka nemithambo iso "Antistius" kunceda ukubuyisela umsebenzi yamehlo retina.
Kuphela inani elincinane amatyala, xa usebenzisa ichiza "Antistius" (kubandakanywa analogs), ngethuba unyango lwesifo sentliziyo, ukusebenza phantsi kuye kwaphawulwa. Mhlawumbi, oko kwenzeke ngenxa yokuba ukuqhubela phambili kwesifo okanye phambi izifo zentliziyo ezingapheliyo.
Kakade ke, wonk 'kufuneka bazi ukuba ukusetyenziswa "Antistius" akuyi kuchaphazela okanye ukuphelisa ukuhlukunyezwa iinkqubo sentliziyo ethukile. Eli chiza wenza kuphela nje inkxaso kunye iindlela zenkxaso. Ngamanye amaxesha oogqirha nokuba amathandabuzo malunga imfuneko yokusetyenziswa kweziyobisi zohlobo efanayo, njengoko kudla izigulana umnikazi ulibale utshintsho, ukuthatha kude kwirejimeni. Noko ke, xa izigulane ukuthobela yonke igqirha ngokuphatha, kwaye ngenxa ALS ngakumbi kwiimeko ezininzi ujika kwagqama evumayo.
Ngoko ke, ukuba sisebenzisa "Antistius" (kubandakanywa analogs) njengoko ichiza ephambili ekulweni ischemia intliziyo, ungafumana japan encinane. Noko ke, ngobuchule ichiza iyazalisekiswa, ukuba asetyenziswe kunyango indibaniselwano njengendlela sokuphucula nethe zeselula. Izigulane basafunda iziphumo zalo, xa kuthelekiswa kunye namachiza afanayo, ithuba lokuba bafunde endaweni yawo kwaye izame ukumisela yeyiphi kakuhle kwaye ikhuseleke ngakumbi?
Ngaphambi kokuba usebenzise amayeza kufuneka udibane nogqirha. Kodwa amava phakheji nganye kukho iziyobisi "Antistius" umyalelo manual. Ukuphononongwa, oogxa bethu ziye ziqwalaselwe ngokweenkcukacha.
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