Zempilo, Amalungiselelo
"Helpeks antikold": imfundiso (tablets). Izimo kunye neziphumo ebezingalindelekanga ichiza
Phakathi izifo egazini SARS kunye neengcaphephe umkhuhlane ingqalelo kakhulu eqhelekileyo. Phantse zonke, kube kanye bejamelene nezi zifo. Okulandelayo, cinga ezimbi ngokufutshane ethile, kwakunye enye amayeza mihla emiselweyo unyango lwabo "Helpeks Antikold" (tablets).
Inkcazelo zokudala kunye nomkhuhlane (short)
Nezifo ezi ezimbi bakholisa ukuba eze kule ngqele. Ngenxa yoko, malunga ne-15% abantu abagulayo ehlabathini. Umkhuhlane - isisifo esibi wentsholongwane egazini zohlobo esosulelayo. Ngaphandle unyango ngokuchanekileyo nangexesha yale ngezifo kungakhokelela ekubeni iziphumo vuhlayiseki kunye nokufa. Umkhuhlane ichaphazela bronchi enkulu kunye noqhoqhoqho. Esi sifo luphawulwa letyhefu kakhulu. usuleleko ezihlasela zosulele ngokuphefumla evusa a ukukhohlela, umqala obuhlungu, icesina kunye intloko ebuhlungu. iimpawu ezifanayo ihambe kunye nomkhuhlane. Omnye amachiza aqhelekileyo olusebenzayo ke ezimbi ingqalelo ithathwa arhente "Helpeks Antikold" (tablets). Izimvo kumagqirha abonisa impumelelo eliphezulu ichiza ngenxa isiphumo entsonkothileyo. Ngokutsho kweengcali, ichiza ngokukhawuleza ngokwaneleyo iququzelela iimpawu zale sifo. Kwi indlela yokusebenza kwezinye iinkcukacha ixelela iqhotyoshelwe kwiziko "Helpeks Antikold" (tablets) myalelo. iingcali Guest alatha ukhuseleko kwemali kunye nonyamezelwano eyanelisayo zezigulane.
iipropati kwemithi
Lithetha "Helpeks Antikold" (tablets) ingxelo ichaza njengoba kulungiselelwa ezintsonkothileyo. Eli chiza iintlungu kunye nesiphumo antipyretic. Kukho kwakhona anti-ezithintela ukosuleleka kunye antiallergic ukusebenza wobulali. Njengoko sinokungqinelwa eqhotyoshelwe kule mali "Helpeks Antikold" iipilisi umyalelo ukunceda ukuphelisa intloko ebuhlungu, amehlo alilayo, ukuxinana ngeempumlo, ukhohlokhohlo. Xa yonyango medicament kuphucula imeko jikelele eziphilayo.
pharmacodynamics
Amalungiselelo iquka amacandelo esebenzayo ezifana phenylephrine hydrochloride kunye cetirizine, kunye paracetamol. Yokugqibela antipyretic, iintlungu kunye nowobulali isiphumo anti-ukudumba. I-paracetamol uyakwazi ukuphembelela iziko thermoregulatory kule ngxenye, zinqanda (zinqanda) kwi Yindibanisela yabalamli ukudumba (serotonin, kinin) kunye prostaglandins. Kunye nale candelo esebenzayo konyusa inqanaba uvakalelo intlungu. hydrochloride Cetirizine kugqalwa womelele ngokwaneleyo antihistamine. Eli candelo ke ochasene akhetha H1 receptor. Ngenxa yayo deceleration umsebenzi gistaminoposredovannoy kwenzeka Isigaba sisandula uxabane nawo. hydrochloride Cetirizine kunciphisa yokufuduka eosinophils kunye nokusasazwa mediators arhabaxa. Ngenxa yoko ke, luyancipha indlela emva kwexesha nawo. hydrochloride Cetirizine uye phantse nafuthe kwezinye ii-. Kule nkalo, oko akuthethi ukubangela antiserotoninovym kakubi kunye neziphumo anticholinergic. phenylephrine Gidrohhlorid udlala uyakhetha udibaniso lwe-agonists. Ngenxa isiphumo vasoconstrictor yababephethwe licandelo esebenzayo, wehlise ukudumba ngeempumlo isifo kunye nesixa imfihlelo eyabelwe. Ukuze ngokwenjenjalo kuphuculwe ukuphefumla ngeempumlo, yaququzelela indlela umoya.
Pharmacokinetics
I-paracetamol ezabalazela ngokufanelekileyo ngokukhawuleza ukusuka kwinkqubo yokwetyisa. Le xi eliphezulu wabona plasma emva 10-60 imiz. Eli candelo isasazwa ngokukhawuleza kwizihlunu zomzimba. Xa kusetyenziswa ngeedosi yesiqhelo kwezonyango, inxalenye encinane kuphela (malunga 28-50%) ka-paracetamol lu dityanisiwe njengeprotini. Kwisiqingatha wobomi - Iiyure ezi 1-3. ixesha effect iintlungu - malunga 4-6, kunye antipyretic - malunga 6-8 iiyure. Nethe ubukhulu becala iiseli esibindini. I-paracetamol iyekelela nkqubo ikakhulu sezintso ngohlobo conjugates sulfate kwaye glucuronic ku-kuwe. Ngaphantsi kwe-5% salawo ingatshintshwanga. Cetirizine hydrochloride kwakhona ako ngokukhawuleza ukusuka kwinkqubo yokwetyisa. ekudleni akuthethi ukunciphisa ivolyum, kodwa kunciphisa kancinane izinga ukufunxeka. Le xi liphezulu icandelo kwi-plasma waphawula emva kangangesiqingatha seyure xa usebenzisa-10 mg. Kukhuthaza cetirizine wenziwa ngakumbi umchamo ngohlobo unmodified. Xa izigulane nokulolonga okanye wobulali umsebenzi othile sezintso kwisiqingatha-ubomi olwandisiweyo iiyure 19-21. Malunga nama-90% kwe candelo ubophelela kwiiproteni plasma. Phenylephrine hydrochloride ako ngokukhawuleza, kodwa ngenxa nethe olukhulu presystemic (ubukhulu becala etorotsitah), bioavailability yayo ngenkqubo malunga ne-40%. Emva kokufumana idosi konwaywa xi ubuninzi saphawula iyure kweeSPU okanye ezimbini. Plasma isiqingatha ebomini ku ezahlukene iiyure 2-3. Emva ukufakwa kwenzeka olunzulu biotransfomatsiya phenylephrine sisibindi. Kukhuthaza kwenzeka ubukhulu becala kusetyenziswa i-izintso ngokohlobo iimveliso yokubola. Ngaphantsi kwe-20% ngesi ifomu kutshintsha.
Iimpawu "Helpeks Antikold" (tablets)
Ukususela oko kunceda eli yeza? Kuthethwa yonyulwa unyango kwangumqondiso influenza kunye izifo ezihlasela zosulele ngokuphefumla egazini, nzima komzimba syndrome. Ezi ukufundwa uqinisekise kwaye ziqhotyoshelwe apha kule medicament "Helpeks Antikold" (tablets) myalelo. iingcali Guest lubonisa ukuba unyango maluqale xa uphawu yokuqala ngezifo. Unyango kwangoko iqale, kokukhona kuya kuthatha inkqubo impiliso.
balawule
Ukwamkelwa kufuneka kwenziwe njengoko abuyise kunye nemveliso "Helpeks Antikold" umyalelo. Iipilisi babelwa izigulane ukusuka kwiminyaka eli-12 ubudala. Izikali - 1 pc. 4 p. / Day. Izigulane ezininzi ukubuza: "Mna macwecwe ezibhaliweyo" Helpeks Antikold "ixesha elingakanani ukuze bawuthabathe.?" Ubude unyango ngamachiza akuntsuku zingaphezu kwe-5. Phakathi amathamo kuyimfuneko ukugcina kudluliswe iyure 4. Kuthethwa asele iyure emva kokutya. Kufuneka ahlambe phantsi kwamanzi ezininzi. Apha imveliso "Helpeks Antikold" (iipilisi) lithethelela ukuba umyalelo umthamo, ukuqeshwa kagqirha. Ukuba akukho isiphumo akufuneki kugqithisela. Kulo mzekelo, kufuneka ubone yincutshe. Ukuba kuyimfuneko, ugqirha angamisela lichiza eyahlukileyo endaweni lithetha "Helpeks Antikold" (tablets). Analogs arhente (iziyobisi "Antigrippin", "Aksagripp", "Antiflu", "Coldrex", njalo njalo) kufuneka zikhethwe kuphela specialist.
Ngubani na akunconywa isixhobo?
Xa Elungiselela "Helpeks Antikold" (tablets) Izimo zezi zilandelayo:
- hypersensitivity ngamnye ukuya amacandelo.
- Kwegazi.
- Hyperthyroidism.
- ngezifo sentliziyo.
- Zisanyisa.
- Ukukhulelwa.
- Iminyaka ukuya kutsho kwiminyaka eli-12.
Ezi zithintelo eziziintloko inikezela ngokusebenzisa "Helpeks Antikold" umyalelo. Tablets kwakhona kucetyiswa ngaxeshanye yeQela tricyclic okanye MAOI.
effect side
Amayeza kungaba nefuthe elibi ekusebenzeni kwenkqubo sentliziyo. Ngokukodwa, kusenokubakho ukuncipha okanye ukwanda koxinzelelo, palpitation. Kwakhona kusenokwenzeka tachycardia. Kwezinye izigulane, kungakhona ukuphazamiseka kwenkqubo womchamo. Ngokukodwa, ekwenzeni "Helpeks Antikold" (tablets) (umyalelo manual iqulathe ulwazi) ingadala spasm we bile wokuchama okanye sphincter vesical. Unyango kudityaniswe opiates kunokubangela nokugcinwa nomchamo. Imithi okulalisa, kungabangela ukozela, lokuqonda luzizi, ukungakhathali, silale, intloko ebuhlungu. Uthomalaliso bangase ngezimvo yokusebenza ngokwasemzimbeni nasengqondweni, ongase, ukungaboni, cinca-cinca, ixhala. Ezi ziphumo bezingalindelekanga zihlobene ukuphazamiseka le CNS. Ngokutsho iingcali, bona ukususela obugqithisileyo idosi konwaywa medicament kuvuka. Ichiza ungabangela ukuba umsebenzi inkqubo yokwetyisa kwamcaphukisa. Ngokukodwa, uthomalaliso sinokufumana kabi esiswini okanye amathumbu, owomileyo umlomo, ugabhe okanye isicaphucaphu. An uxabane iquka irhashalala.
oyi
Njengokuba ekhankanywe apha ngasentla, ukuba ziqhubeka, udibane nogqirha. Kufuneka kutyelela oyingcali kwimeko sufaka kubonakaliswa ngezifo. Ukongeza kule umda ngentla, kukho ezinye iimeko apho kufuneka uqaphele kakhulu. Olu luhlu luqulethe eqhotyoshelwe kule medicament "Helpeks Antikold" umyalelo. Tablets, ingakumbi, ngononophelo kakhulu izigulane kakuhle kwezintso okanye umsebenzi hepatic. Ngexesha unyango, ithamo kufuneka kungagqithwa. Kwakhona, musa uthathe amanye amayeza, njengenxalenye apho kukho paracetamol. Amathuba libanda iphezulu kakhulu izigulane netsirroznymi isifo sesibindi, nomsindo kakubi utywala. Isilumkiso kuyafuneka ukuqeshwa ichiza ukuba izigulane seswekile, kwakunye neglaucoma engile-ukuvalwa. Kufuneka kukhunjulwe ukuba felilefrin sikwazi ukwandisa uxinzelelo. Kulo mba, kusenokufuneka i uhlengahlengiso uwadle izigulane zifumana unyango umfutho, kwakunye beta-adrenergic receptor. Njengenxalenye ichiza "Helpeks Antikold" (tablets) (ifoto beziyobisi linikwa kwi nqaku) iqulethe aspartame. Eli candelo - umthombo phenylalanine. Le ayimbumba ichaphazele imeko izigulane kunye phenylketonuria. Kufuneka ubeke ichiza ukuba izigulane ezinqabileyo ilifa ukunganyamezelani fructose, sucrase-isomaltase imibala, ngokunjalo malabsorption glucose-galactose.
Ukukhulelwa ne zisanyisa
iziphumo zophando eyaneleyo esalatha ukhuseleko ukusetyenziswa kwemali "Helpeks Antikold" ngexesha la maxesha apho. Kuye kwafumaniseka ukuba phenylephrine kunye paracetamol uyakwazi ukungena kwi ubisi. Kulo mba, amayeza "Helpeks Antikold" ngexesha zisanyisa ayivumelekanga. Ukuba kuyimfuneko, unyango kule zokuxheshisela thuba kufuneka kupheliswa.
Ukuze ufumane inkcazelo engakumbi,
Eli chiza ingenza ukozela, ukungaboni kunye nezinye izifo CNS. Kulo mba, kuba ixesha lonyango, izigulane kufuneka uyeke izinto ezinokuba yingozi. Ingakumbi kumayelana abaqhubi kunye nabo yokusebenza enxulumene iindlela kwaye ufuna eliphezulu yoxinaniso ingqalelo kunye quickness esizenzayo lengqondo. Ukusebenza kunye nokhuseleko izigulane abangaphantsi kweminyaka eli-12 ubudala iye ayasekwa. Ngokuphathelele olu nyango "Helpeks Antikold" izigulane kweli qela lobudala akayi wabelwa.
intsebenziswano
Lithetha "Helpeks Antikold" kufuneka abasayi kwenziwa kubanjiswene ne-Mao inhibitors Yolule iiveki 2- emva kokuba ulwamkelo zabo. Akunconywa amayeza ngaxeshanye kunye namanye amachiza eziqulathe acetaminophen, kwaye zilungiselelwe yonyango uxinezeleko, isifo Parkinson ngayo, ukuphazamiseka engqondweni. arhente ukusebenzisa ixesha elide "Helpeks Antikold" ngoyo isiphumo ichiza "Warfarin" kunye nezinye coumarins. nomthelela obonakalayo ibonakele unyango uveza. Kunye kunye nokwamkelwa lithetha "Helpeks antikold" a medicament "Cholestyramine" uyancipha absorbability yaye iphungula sisenzo paracetamol. Ukwandisa kukufakwa icandelo amachiza afana "Domperidone" yaye "metoclopramide". Xa isicelo ngokudibene NSAIDs kwandisa amathuba lomonakalo kwezintso. Umngcipheko lweziphumo eziyityhefu kunyuswa unyango ezihamba kunye iziyobisi ukwandisa umsebenzi enqanda zesibindi. Ezi ikakhulu ziquka barbiturates, iziyobisi antiepileptic kunye namayeza "Rimfampitsin". Medicine "salicylamide" kwandisa isiqingatha-ubomi paracetamol. imiphumela Hepatotoxic ngabaya ukuba mandundu ukusetyenziswa emanyeneyo ichiza "Helpeks Antikold" baligalele.
libanda
Xa ezibanjiswe mali ye zonyango kunene kwaye yanika ubukho imiba emayezeni paracetamol ukusebenza hepatotoxic. Emva chemical libanda, kunye nokwenzakala wesibindi lwezonyango waphawula emva kweeyure 12-48. Olunye lweempawu zokuqala sibizwe ngokuba blanching ulusu, iintlungu esiswini, ukugabha kunye isicaphucaphu, unesifo. A ingozi ephezulu ezingaqhelekanga inkqubo glucose ukutya kunye mhlawumbi ne-asidi eninzi. Amatyala pancreatitis kunye arrhythmias akhawunti in practice. Mhlawumbi njengokuba necrosis wesibindi, nezintso glomeruli. Kwimeko libanda inokuphuhlisa thrombocytopenia, wasondela kwikhoma hypoglycemic. ukozela Ukwanda xa efumana isixa esikhulu medicament kungenxa yesenzo cetirizine. Ngelo xesha abantwana excitation lokuqala kwenzeka, ngoko enika indlela eya bengenamdla. Xa libanda, nokuba imeko eqhelekileyo yempilo zibhekisela ingcali ngokukhawuleza kangangoko kunokwenzeka.
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