Zempilo, Amalungiselelo
"Artrokol" (gel): imiyalelo ukusetyenziswa, analogs kunye nohlolo
Ndingayisebenzisa njani ichiza "Artrokol" (gel)? Imiyalelo zokusetyenziswa ichiza ziza kuchazwa kweli nqaku. Kwakhona, uya kufunda koko iyeza emiselweyo kwizigulana, nokuba unawo analogue, kunye nazo naziphi na izimvo malunga seliphumile nkonzo.
Imixube, iziyobisi ezingxobeni nemilo yayo
"Artrokol '- gel (2,5%) ukwenzela ukusetyenziswa lwangaphandle. Ekuthengisweni ifike kwi-aluminiyam ityhubhu 45 Kwakhona kwi ibhokisi yekhadibhodi kunye ichiza nephetshana imiyalelo eneenkcukacha ukusetyenziswa.
Oko iqulethe ichiza lwangaphandle "Artrokol" (gel)? 100 g kwesi eziqulethwe 2.5 g lwe isithako esebenzayo, njengoko ketoprofen. Ngaphezu koko, eli chiza phantsi ingqalelo ibandakanya ezi zinto inkxaso ilandelayo: trolamine, Carbomer 980, 96% ethanol, ngamanzi okuhlamba kunye methyl parahydroxybenzoate.
Umgaqo ekusebenzeni medicament
"Artrokol" - ijeli, eyona nto esebenzayo yenziwe ketoprofen. Wathi medicament ngamalungu kwiqela amachiza nonsteroidal anti-ukudumba, kwakunye avela of arylpropionic acid.
medicament izinto Base ingqalelo inika isiphumo anti-ezithintela ukosuleleka kunye iintlungu, olwenzeka ngexesha inhibition non-uyakhetha of Cox-1, bradykinin kunye Cox-2, kunye inwebu uzinzo (lysosomal) kunye inhibition of macrophage yokufuduka.
Ukongeza, iziyobisi "Artrokol" (gel) ebonisa izinto anti-ukudumba kunye iintlungu. Iyakwazi ukwenza kwiseli kwisigaba nemithambo phambi kwexesha nasemva kwexesha inkqubo arhabaxa. Kwakhona, eli chiza ehla zegazi udibaniso.
Ezona mpawu pharmacokinetic of
Ngokutsho imiyalelo eqhotyoshelweyo, ketoprofen (isithako esebenzayo ye medicament) emva kokuba isicelo mlonyeni nolusu ako, uze emva koko lingena singene embindini inkqubo yokukrala nangexesha ixesha elide ugcina i olifunayo xiyimiso kwezonyango emzimbeni.
Kukufakwa ichiza waya kuye kwasasazwa ngenkqubo minimal (5% of ithamo esetyenzisiweyo). Kulo mzekelo, ukufunxeka kumlanjana igazi olucothayo kakhulu.
Uyondelelwano lwee- isithako esisebenzayo beziyobisi (usebenzisa 50-150 mg of ketoprofen) egazini emva kweeyure 7.5 yi mg 0.08-0.15 kuphela / ml.
Drug "Artrokol" (gel) kunye nenjongo yawo?
Le zibonisa ukuba ukusetyenziswa ijeli ethathelwa ingqalelo ukuba lithi zilandelayo:
- myalgia, rheumatism kunye rheumatism imvelaphi;
- izifo kwenkqubo musculoskeletal (kuqukwa isifo samathambo, syndrome articular ngexesha exacerbation sifo, ankylosing spondylitis, samathambo psoriatic, osteochondrosis, osteoarthritis of eyendawo ezahlukeneyo, sisilonda esidumbileyoesingaphakathi yokukrala imisipha, nemisipha, sciatica, bursitis okanye lumbago);
- njengenxenye yonyango leqela le ukudumba ezimbi imithambo (umz, phlebitis, periphlebitis), iindawo nkovu okanye iimpahla nkovu (umz, lymphangitis, lymphadenitis phezulu);
- ukudumba post-traumatic kwenkqubo musculoskeletal kunye kwizihlunu ezithambileyo (kuquka unyango kwangumqondiso yokwenzakala ayinzima, kuquka komsipha, ukwenzakala ezemidlalo, komsipha okanye iinyembezi zabo imisipha kunye nemisipha, nemivumbo, iintlungu post-traumatic).
Siphelisa ukusetyenziswa
Ntoni "Artrokol", linamafutha aqholiweyo kunceda, siye ezichazwe apha ngasentla. Noko ke, oku kuthetha ukuba kukho Izimo. Ezi ziquka oku kulandelayo:
- ababudala bungaphantsi kweminyaka 12;
- uvakalelo oluphezulu ukuya iziqalelo neziyobisi kunye acetylsalicylic acid kunye nezinye NSAIDs;
- senyanga yesithathu yokukhulelwa kunye nokuncancisa.
Drug "Artrokol" (gel): imiyalelo yokusetyenziswa
Kuba unyango enye yejeli ingakhulula 5.4 cm phantsi ingqalelo kuthetha isicelo isikhumba kwindawo ezifunwayo kunye kuzonwaya ethambileyo umphululela iintshukumo de ukufunxeka kwayo ngokupheleleyo.
Kufuneka kuqatshelwe ukuba ezinkulu ummandla kummandla ochaphazelekayo, kokukhona ichiza ingena yenkqubo yonyango. Ngaloo strip pyatisantimetrovym medicament "Artrokol" ingqamana 100 g ketoprfena.
Emva kokuba kusetyenziswa neoli, kufuneka ngoko nangoko uhlambe izandla.
gel kujongwa uvumelekile ukuba asebenzise ngokubambisana namanye imithi equlethe ketoprofen (umz, libambisene kunye emacwecweni, njengezingxobo, suppositories efakwa).
Ithamo ubuninzi arhente yi 200 mg ngosuku. Esi sisixa ichiza akuxhomekekanga kwindlela amayeza.
Ixesha le khosi unyango kufuneka kumiselwa qho ngamnye ngugqirha khona. Nakuba kunjalo, kufanele kuqatshelwe ukuba liniment ukusetyenziswa iintsuku ezingaphezu kwe-10 ilandelelana akuvumelekanga.
ziphumo bezingalindelekanga kunokwenzeka
Yiyiphi imiphumo emibi kunokubangela ichiza "Artrokol" (gel)? Imiyalelo uthi malunga imiphumela emibi ilandelayo yendalo:
- bronchospasm, angioedema;
- ukuhlaselwa somoya, reactions anaphylactic kuquka ukothuka;
- ububomvu, ukurhawuzelela, irhashalala, avuthayo, ukudumba kwesikhumba;
- nangokhwekhwe phlyctenular bullous nabanako wokusasaza kwezinye iindawo ukuze ufumane ngokubanzi;
- photosensitivity, bullous okanye xhumana dermatitis;
- isicaphucaphu, Stevens-Johnson syndrome, ukugabha;
- ukopha, izilonda esiswini, urhudo, heartburn, ukuqhina;
- Disorder umsebenzi kwezintso, exacerbation ukusilela indalo esingapheliyo kwezintso, nephritis Embi kunye ukusilela kwezintso.
Kufuneka kuqatshelwe ukuba xa usebenzisa gel "Artrokol" kungabangela ezinye reactions icala kunye nenkqubo yokucola ukutya kunye nenkqubo womchamo. Ubunzulu ezi ziphumo kuxhomekeke kwimali iziyobisi kunye nokukwazi irhasi zithako yalo, indawo baphathwa ubungakanani, umyinge kunye nexesha imeko zonyango kwesikhumba.
Asinako ukuba abantu abadala sihlaselwe yeziphumo ezibi ze NSAIDs kulo unyango.
Ngethuba lokukhulelwa zisanyisa
Ngaba ukusebenzisa iziyobisi "Artrokol" (gel) ngethuba lokukhulelwa nokuncancisa? Ekuhambeni-experimenti kwi namabuzi, kwaye kwafunyaniswa ukuba imali akuthethi ukuba isiphumo yaManzi naMahlathi kunye embryotoxic ezilwanyaneni abaselula. Nakuba kunjalo, kufanele kuqatshelwe ukuba sisiphumo esincinane embryotoxic kuye kwaphawulwa ukuhlola kwi imivundla.
Ekubeni ukhuseleko ketoprofen kwabasetyhini abakhulelweyo khange yaxhaswa naziphi na izifundo, iingcali musa yaleza ukusebenzisa esi sixhobo koomama abakhulelweyo.
Kwakhona kufanele kuphawulwe ukuba ketoprofen kunye nezinye inhibitors of prostaglandin amagama kungabangela zinetyhefu sezintso, yemiphunga nezengekho neenkqubo kwentliziyo yosana olungekazalwa.
Iimveliso kuwohloka mali afumaneka ngobisi lwebele. Ngenxa yesi sizathu, eli gel "Artrokol" akumele kwenziwa ngabo nursing abafazi.
ulwazi oluthile
Ukulungiselela "Artrokol" (gel), apho analogs zidweliswe ngezantsi, oko aluvumelekanga isicelo kwiindawo ulusu kunye notshintsho zophendlo lwezifo ezifana induna okanye onokhwekhwe. Kukwasebenza kwanjalo kuyo kummandla abosulelekileyo okanye amanxeba avulekileyo.
Kufuneka kwakhona sikuphephe qha kweziyobisi kunye ngenwebu yangaphakathi. Emva ngokusebenzisa ichiza kufuneka ahlambe izandla zabo.
Esi sixhobo ayikho alungele ukusetyenziswa kunye zokubopha occlusive.
Ngexesha unyango "Artrokolom" kwaye iiveki ezimbini emva kokuba kunyango, kungakuhle ukuphepha udibana nesikhumba elangeni ngqo.
"Artrokol" (gel): ncomo kunye amalungiselelo ezifanayo
Ngu analogue kweli chiza ziquka iziyobisi ezifana "Karmolis-gel", "Indomethacin", "diclofenac", "Remisid", "Vipratoks", "Denebola", "Injongo yale T", "chondro-amandla", "ibuprofen" "Ketonal" kunye nabanye.
Yintoni abantu bathi abasebenzisi iziyobisi ngayo? Bathi gel "Artrokol" imele i-arhente olusebenzayo anti-ukudumba. Iziphatha kakuhle ezo iimeko zophendlo lwezifo ezifana myalgia, izifo inkqubo weentshukumo, izifo yokukrala imithambo, nangokurhala post-traumatic.
Bobubi yalo amayeza isicelo lwangaphandle zibandakanya nobuninzi icala elingenzi nto-leyo azibonakali emva kokusetyenziswa gel. Kaninzi, izigulane kuvandlakanywa ukuba bomvu, ukurhawuzelela, izigxala, ukutshiswa kunye ekweneni eluswini, kwakunye isicaphucaphu, nangokhwekhwe, izilonda esiswini, urhudo kunye heartburn. Enye engxakini ichiza kuqwalaselwa kukuba akukho emiselweyo ukuba abasetyhini abakhulelweyo, kwakunye nokusetyenziswa ngexesha zisanyisa.
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