ZempiloAmalungiselelo

Imiyalelo isicelo, ingxelo kunye analogue "Locri"

isifo sentliziyo unesifo kuxhaphakile kakhulu ehlabathini. Esi sisifo noko obufihlakeleyo, esemfuleni isaqala kunzima ukuchonga. Ngoko ke, emva kweminyaka engama-40, kufuneka iliso dvleniya yokusebenza rhoqo. Ukuba iziphumo ziphezulu kakhulu, kufuneka udibane nogqirha wakho. Kokuqala unyango kwangoko, i ngokukhawuleza unako ukuyoyisa le sifo.

Amachiza Modern luphawulwa kahle eliphezulu. Eli qela blocker. Tablets kakuhle kakhulu kuthoba uxinzelelo lwegazi kwaye musa ukulimaza umzimba. athandwa kakhulu phakathi zeetheraphisti namhlanje ukulungiselela "Lokren". Imiyalelo yokusebenzisa, analogs, idosi echanekileyo - yonke le nkcazelo ithiwe thaca apha ngasezantsi.

Ukubunjwa kunye nefomu yokhululo iziyobisi

Tablets "Lokren" emhlophe, khaxa kancinane kwicala elinye ephawulwe nombhalo EK20. Ekubeni titer enjalo amayeza zingahlukaniswa ngokulula ukusuka mbumbulu. Amacwecwe anxibé kwiqokobhe obhityileyo. Icandelo iphambili ekwakhiweni kwezi tablets ithathwa gidrohrorid betaxolol mg-20. Nezincedisi machiza monohydrate lactose, neselulosi kakhulu, sodium karboksilmetilkrahmal.

Iqokobhe ubunjwe gipromilozu, macrogol, titanium dioxide. Ifumaneka iipilisi ngendlela blister, kunye iziqwenga 14 nganye. Nayiphi Togu "Locri" kuya kuba sisincoko efanayo nokubonakaliswa zokusetyenziswa.

Iziphumo ichiza emzimbeni

Iipilisi lilungu kwiqela beta-blocker. Bona zithathwa blocker uyakhetha kumqolo wokuqala. Betaxolol, eyinxenye beziyobisi, ngandlela ukuvimbela beta-adrenoceptor cardioselective, luphawulwa kukungabikho komsebenzi agonist na ndizayo buthathaka. Ngenxa ukuncipha iziyobisi izinga lentliziyo ngexesha umsebenzi lokuphumla ngokwasemzimbeni. Iimpembelelo eziphambili - kunciphisa uxinzelelo igazi ukuphumla nasebudeni umthambo.

Xa usebenzisa ichiza udlula tachycardia, kunciphise umthwalo entliziyweni, eqhelekileyo yoluvo nokuhamba kwegazi. umfutho of betaxolol kunye nokusetyenziswa ixesha elide akukho lifinyele. Xa elinye yokufakwa idosi emacwecweni lawo isiphumo enyangayo kwenzeka kwisithuba seeyure ezintathu kwaye iqhubeka yonke imihla. nemiphumo emihle kunokuzuzwa kunye ikhosi clusive zonyango. Izenzo ezinjalo ziye kwi iipilisi umzimba "Lokren". analogue Drug kwakhona normalizes izikhombisi igazi xa zisetyenziswe ngokuchanekileyo.

Pharmacokinetics

Xa ongena ebantwaneni, ichiza ngokukhawuleza iyachithakala kwaye 100% etsalwe esiswini. Isiphumo esiphezulu ifunyanwa emva kweeyure ezimbini plasma. Ichiza enebana ubonelelo igazi ngama-50%. Betaxolol in esibindini wakha metabolites engasebenziyo. Phantse 80% ze eyona nto esebenzayo idubule yi izintso eluhlobo metabolites. 20% ivela emzimbeni ingatshintshanga.

Akakhawulezi ngokwaneleyo kunokwenzeka ukuba kuzuzwe iziphumo ezihle unyango, ukuba uthathe iipilisi "Lokren" ngokufanelekileyo. Imiyalelo yokusebenzisa ezinayo yonke ingcaciso eyimfuneko.

Iimpawu kunye Izimo

Isizathu yokuqeshwa ichiza uthathwa lwegazi. Iindlela singathathwa wedwa okanye zidityaniswe namanye amayeza ukuba azole ukuhlisa uxinzelelo. Iipilisi sabelwe khona ukuze kuthintelwe imivumbo e.

Izimo kunyango ngamachiza kucingwa isifuba inyumoniya kakhulu kwaye kwemigudu yomoya, ukusilela intliziyo oyingozi. Musa ukuthatha iyeza kwi wavakalisa nesenzeko bradycardia, iintlobo okunzima sisifo Raynaud kaThixo kunye ukuphazamiseka neuropathy kwegazi. Kukho imida yobudala. Amayeza engamiswanga izigulane ezincinane.

Ayikhuthazwa ukusela iipilisi kwizigulane kunye insufficiency kwezintso okanye hepatic. Ngethuba lokukhulelwa isixhobo lokwaphusa zingasetyenziswa kuphela xa inzuzo engase ukuya unina komonakalo ezinokuba nobungozi usana.

Phambi unyango kufuneka ufunde ngenyameko imiyalelo malunga nokusetyenziswa kwemali "Lokren". iingcali Guest lubonisa ukuba iziphumo ebezingalindelekanga akholisa ukubakho kwabo izigulane abangawuthobeliyo izindululo.

balawule

Ichiza kufuneka athathwe yindyebo iziselo. Iyeza kufuneka ukuhlafunwa. Unyango kufuneka luqale ioli esisiqinqatha icwecwe (10 mg). Ukuba nempembelelo entle unyango, kubalulekile ukuba ukwandisa umthamo akayi kuza iiveki ezimbini. Izinga eliphezulu ngemihla ayikwazi ngaphezu-40 mg.

Oogqirha abaninzi azilukhuthazi kwizigulana abo ukuba basele ipilisi ngaphezu kwesinye ngosuku. Ukuba unayo zokucutha ihlwempu kuyimfuneko ukuba ongeze omnye unyango ngamachiza umfutho. Izigulane insufficiency kakhulu sezintso kufuneka uqale ukuthatha amachiza ithamo of mg-5. Ngcembe ukunyusa izinga ngemihla. Limelwe ukuba kufundwa phambi kokuba kusetyenziswa iindlela "Lokren" umyalelo manual.

libanda

Ngenxa libanda, iipilisi zinokuba vertigo, drop nehigh, cyanosis leminwe nezikhonkwane, bradycardia, lightheadedness. Kwakhona nezimpawu ezifana bronchospasm kunye nokungaphumeleli intliziyo.

Unyango libanda yenziwa lavage esiswini. Kuyanconywa ukuba asele adsorbent nomonde ezidityanisiweyo nonyango nokubandakanywa. Xa ukuhla xi kuyimfuneko ukuba prokapat "Dopamine" kwaye ngenisa "Atropine". Kufuneka ngokuqinisekileyo ukongeza glycosides intliziyo kunye antispasmodics. Kwiimeko kakhulu, loo nto ibonisa ukuba kuqaliswe ababambeleyo igazi plasma. Nayiphi Togu "Locri" kufuneka, emva idosi emiselwe ngugqirha.

imiphumela emibi

Xa ukuphatha ungakwazi ukuqala reaction iziyobisi komzimba. Oku kubonakala ngokohlobo kwamaqhakuvana kwi ulusu kunye ukulunywa. Kwakhona, kukho reactions kwicala e-nervous system, apho kuboniswa nesiyezi, intloko ebuhlungu, asthenia, sokulibala, amabi, paresthesia. Iziphumo ebezingalindelekanga ziquka lehla umbono, ukunciphisa uxinzelelo intracranial. Ngelo xesha ukuthatha iipilisi zidla wabona iintlungu esiswini, isicaphucaphu, ukugabha. Ngamana ukutshintsha igazi kunye nokuphuhlisa leukopenia. Abantu ezithatha ichiza kubangela induku. Ukuqapha kufuneka kuqeshwa iipilisi ebudaleni.

Kufuneka igcinwe kwiqondo lobushushu igumbi kwindawo emnyama itshixwe abantwana, ichiza "Lokren". Analogs esetyenziswa nemiqathango efanayo.

Togu "Locri" eRashiya - ichiza "Betaxolol"

Indlela ukuba ukhethe indawo esemgangathweni amayeza? Kuthekani ukuba ekhemesti akazange abe indlela 'Lokren "? analogue Drug uya kusoloko kukwazi ingcebiso kugqirha. Popular esebenzisa "Betaxolol." It cardioselective beta-blocker esetyenziswayo ukuthoba uxinzelelo lwegazi kunye nokuhlaselwa angina. Emva kokungenisa lwanamathela ngokupheleleyo esiswini. Isiphumo esiphezulu ifunyanwa kwi plasma iiyure ezintathu. Ichiza kwazona yi izintso ngokohlobo metabolites enziwa esibindini.

Ichiza kwandisa uxinzelelo intraocular kakuhle, ukuba usebenzisa isisombululo ngokohlobo wamehlo.

Iyeza lisetyenziswa kanye ngosuku ngexesha umthamo mg-20. Amayeza zingasetyenziswa yedwa okanye njengenxenye yonyango udibaniso. Akukhuthazwa ukuba zisetyenziswe ngexesha lokukhulelwa kunye zisanyisa. Kwiimeko ezinqabe kakhulu, ichiza ibanga iziphumo ebezingalindelekanga ngohlobo kwamaqhakuvana kunye nokushisa apha esikhumbeni. Kwakhona, kusenokubakho isiyezi kunye isicaphucaphu, kwakunye usebenzisa iipilisi "Lokren". nucleoside Russian abe ebonisa efanayo Izimo.

Drug "Betacam"

Amayeza bobabo beta-blocker kumqolo wokuqala. iipilisi ezimhlophe. ithamo nganye 20 mg betaxolol hydrochloride. Amayeza kungenziwa kumiselwe kuphela ngugqirha. Ichiza inceda bunjani uxinzelelo lwegazi, ukunciphisa izinga intliziyo ngexesha lokuphumla kunye ngexesha umthambo, oko kukhokelela eziqhelekileyo peripheral kwegazi nokuphelisa angina.

Akukhuthazwa ukuba amayeza e ezimbi ze izintso wesibindi. Ngethuba lokukhulelwa lokwaphusa ichiza akuvumelekanga. Wezindlu baxabane nomzimba kunye ezinxaxhileyo okuncinci iinkqubo luvo esiswini. Amanyathelo kufuneka umiselwe abantu ebudaleni kwaye kwimeko hypersensitivity ukuya amacandelo amacwecwe. Le Togu "Locri" buyisela ngokupheleleyo original amazwe.

reviews

Malunga Beta-blocker ziingcali ukuthetha kakuhle. Kuba ixesha elifutshane kunokwenzeka bunjani parameters kuxinzelelo kunye nokunciphisa ventricular hypertrophy ekhohlo. Ezi Amachiza ukunyamezeleka kakuhle kwaye aluchaphazeli umsebenzi namanye amalungu kunye neenkqubo. Nayiphi Togu "Locri" iya kubonisa nemiphumo emihle ukuba isetyenziswa ngokungqinelana nemiyalelo.

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