Zempilo, Amalungiselelo
Ichiza "Relakson": imiyalelo ukusetyenziswa, inkcazelo, izimvo, analogue
Ziziphi yedosi emiselweyo ichiza "Relakson"? Imiyalelo malunga nokusetyenziswa kweziyobisi kuya kuxoxwa ngezantsi. Kwakhona, uya kufunda malunga kukuba ingaba olu nyango analogs kufuneka, wobeka phi kubiza, apho kunokwenzeka khona ukuba kuboniswe, njalo njalo. D.
Imilo, inkcazelo, ukwakhiwa kunye nokupaka
Ukulungiselela "Relakson" evela ngokohlobo amacwecwe biconvex ngeenxa emhlophe umboniso-camera. Eyona nto elikhutheleyo ichiza zopiclone. Kwakhona medicament iquka excipients zilandelayo: hypromellose, microcrystalline kwincindi, lactose, iitapile starch colloidal lesilicon dioxide, talc, isodiyam carboxymethyl starch, povidone, macrogol, nemagnesium stearate kunye titanium dioxide.
Xa iphakheji uthengiswe "Relakson" tablet? Imiyalelo ukusetyenziswa livalelwe yimfumba yekhadibhodi, neziwela kwaye aya esiseleni kunye ichiza.
iimpawu pharmacodynamic
iziyobisi "Relakson" Zisebenza njani? Imiyalelo yokusebenzisa ingxelo yokuba eli thile ngoweqela tsiklopirrolona qela. Ngokwemo, kuba kwahlukile barbiturate kunye benzodiazepine hypnotics. Le ichiza a agonist benzodiazepine receptor. Yokuxoxisana nabo, ukuba akayi kungena ukudibana kunye nezamkeli peripheral.
iimpawu ichiza
Yintoni iimpawu iyeza "Relakson"? Iingcali Ukubuyekezwa ingxelo ukuba esi sixhobo unako unenye sine, anticonvulsant thile inobulali, relaxant kwezihlunu kunye tranquilizing neziphumo. Bonke bephela ahlangene ngesenzo receptor Gaba oluntsonkothileyo macromolecular.
Emva kokufumana iipilisi eyomeleziweyo isiphumo inhibitory ka Gaba, kwaye kananjalo zicinezelwa transmission interneuronal kwi CNS.
ipilisi zokulala "Relakson" shortens kakhulu ixesha ubuthongo kunciphisa inani eke ebusuku kwaye kuphuculwe umgangatho ubuthongo. Kwakhona, eli chiza kwandisa ixesha ebuthongweni kunye ngenkankulu ibanga iziphumo postsomnicheskih ezinjengezo ukozela yaye ubuthathaka kusasa.
Habituation kwi intshukumo isimaphambili se ichiza ongekhoyo. Ngoko ke, oko kuthathwa kwindlela ibhetshi ukuya kwiiveki 17.
Le pharmacokinetics beziyobisi
Drug "Relakson", ixabiso yayo eboniswe ngezantsi, ngokukhawuleza wendele kunye neeyure sele emva 2 iqatshelwe egazini. Ukufumana ukutya aluchaphazeli ukufunxeka amayeza. Kwi-45%, Sithe nca kwiiproteni igazi.
Kwanasemva kokuba ubuchule eziliqela kumacwecwe ukuqokelelana lwesiyobisi esebenzayo kunye metabolites zingaphawulwa.
Isiqingatha-ubomi zopiclone kunye metabolites ezinkulu iiyure 7.5 no 4.5, yaye zopiclone lingatshintshanga - iiyure 5.5. Malunga nama-80% ye ichiza idubule kunye nomchamo, kwaye 17-20% - kunye endleni.
abantu abadala iziyobisi yokucolwa esibindini kuyehla. Ngaphezu koko, isiqingatha-umphefumlo wayo kuyoluka iiyure 7. Ngokumalunga nokwanda ukwimo esebenzayo, oko akuyi ukubonwa kwi amacwecwe zedosi ezininzi.
Ubungqina obubonakalayo buxela
Kufuneka wenze ntoni ukuphuthelwa? Oogqirha bacebisa ukuba athathe "Relakson". Le mveliso yenzelwe yonyango ukuphuthelwa ezingapheliyo kunye zezomzuzwana lwemeko abadala. Kwakhona, oku ngenkuthalo isetyenziswa yi abo bangakwaziyo nokulala, Ekuvukeni zasebusuku nasekuqaleni.
Izimo
Tablets "Relakson" akukhuthazwa kwezi meko zilandelayo:
- hypersensitivity kweziyobisi ukuba izinto kwisiseko;
- i kakhulu lwe myasthenia gravis;
- ngexesha lokukhulelwa;
- kunye belele ;
- ukusilela zemigudu;
- ukuhluleka kakhulu isibindi;
- ngaphantsi kweminyaka eli-18.
Drug "Relakson": imiyalelo yokusebenzisa
Ngaphambi ukuthatha ipilisi zokulala Kucetyiswa ukuba udibane nogqirha. Kuyimfuneko ukuba ukufunda imiyalelo apha.
"Relakson" Amacwecwe (igama generic - "Zopiclone"), kuthathwa ngomlomo, nje phambi kokuqala ngokulala ubuthongo. Abadala iziyobisi esebenzayo yaphathwa ne nedosi ye-7.5 mg. Le mali iphezulu yi-15 mg koncedo ubuthongo.
Ubude lilonke ukusetyenziswa tablets akufunekanga ibe ngenyanga ngaphezu kwesinye. Kwimeko nganye, ubude unyango kumiselwa ngamnye ngokuxhomekeke kwimeko yomguli, kunye nohlobo ugwayi.
Thatha amayeza xa ukuphuthelwa ehlala Kuyancomeka malunga 3-5 mihla lwemeko - iiveki 2.5-3. Ixesha lika-unyango ukuphuthelwa ezinganyangekiyo kufuneka kumiselwa kuphela ngugqirha.
abantu abadala kunye ezingapheliyo sisifo obstructive pulmonary, kwakunye nomsebenzi isibindi kakuhle elawulwa 3,75 mg iziyobisi. Ukuba kuyimfuneko, wathi ithamo kufuneka kwandiswa ukuya 7.5 mg.
Unyango lwe ugwayi kwizigulane kunye insufficiency sezintso nazo eqala nge ½ unabo, oko kukuthi, 3,75 mg.
amacala libanda
Ukuthatha amathamo ezinkulu thile ebangela CNS ukudakumba of ubuchule ubucaka (kwi somnolence ngokukhawuleza kwi imeko isiqaqa).
Therapy luqala i lavage libanda esiswini. Okulandelayo, isigulane emiselweyo sorbents.
Kwakhona unyango kwangumqondiso kunye nokuhlolwa kwemisebenzi zomzimba ebalulekileyo. Drug "Flumazenil" kusetyenziswa alikaziwa.
imiphumela emibi
Zintoni iziphumo elicala "Relakson"? Izimvo yeengcali abanamava ingxelo ukuba eli chiza ukuze negalelo kuphuhliso ziganeko zilandelayo:
- isicaphucaphu, kome nobukrakra emlonyeni;
- isiyezi, intloko ebuhlungu, nobuthongo okuncinci kusasa;
- amabi, ukuba ndlongondlongo, ukuba nochuku, nemibono, eziya zisiba of imo kunye zikarhulumente edakumbisayo, kwakunye nokuphuhliswa kunesifo (ezinqabileyo kakhulu);
- ukurhawuzelela, irhashalala, reactions anaphylactic (ezinqabileyo kakhulu);
- transaminases isibindi kunyuswa aze obrak phosphatase.
Kufuneka kuqatshelwe ukuba kwiimeko ezinqabileyo, ichiza ebangela "khansela" syndrome, yaye ngenxa yoko, okuvuka ugwayi.
imithi
Ngoku uyazi ukuba yintoni ezakwenziwe malunga ugwayi. Reception "Relakson" ichiza kufuneka silumke kakhulu, ingakumbi ukusetyenziswa ngaxeshanye amanye amayeza.
Ngokutsho imiyalelo, ukwanda ukusebenza inhibitory kwinkqubo luvo beziyobisi lwenzeka xa zidityaniswe kunye lakhula, neuroleptics, iintlungu, uxinezeleko, nadlamkisayo kunye hypnotics, yaye "Erythromycin" antiepileptic kunye antihistamines, analgesics ezidakumbisayo.
Ayikhuthazwa ukusela utywala kunye namayeza utywala aqulethe ngaxeshanye "Relaksonom". Oku kungenxa yokuba yindibaniselwano loo yandise yayo okulalisa.
Ukufumana amayeza thile kunciphisa kakhulu perfonala xi okanye trimipramina igazi. Oku kufuneka ithathelwe ingqalelo xa ukuqeshwa kwabo ngaxeshanye.
iingcebiso ezithile ngokufumana thile
Into ekufuneka uyazi phambi kokuba uthathe iziyobisi "Relakson" (efana kwesi sixhobo zidweliswe ngezantsi)?
Abantu ukuhlaselwa sisifo sombefu ebusuku zidityaniswe kunye namayeza methylxanthine inani ipilisi zokulala kunciphisa inani kuhlaselwa kwiiyure ekuseni, yaye kunciphisa namandla kunye nexesha.
Xa kunikwa "Relakson" Maze ngokupheleleyo zicime ithuba likhoboka. Kuxhomekeka ingozi beziyobisi lwenzeka kwezi meko zilandelayo:
- waphula lwendlela kunye nobude zonyango;
- kakubi utywala okanye iziyobisi;
- xa kudityaniswe utywala nezinye iziyobisi psychotropic.
Ukwenzela ukuphepha syndrome of "ukurhoxiswa" bayeke ezithatha ichiza kufuneka ngokuthe nokunciphisa umthamo ukuya ubuncinane.
Xa abafumana ipilisi zokulala nomonde bangafumana kunesifo anterograde. Idla kubonakala xa ubuthongo lomncedis, yaye emva kwexesha lekhefu elide phakathi kolawulo iziyobisi kunye lokulala.
Ukunciphisa ubungozi ezinjalo, kuyimfuneko:
- Ubude Sleep ukubonelela iiyure ezi-6;
- ukuthatha amayeza phambi kokuba uye kulala.
amayeza kubhekwe ukuba kuboniswe ukuba unyango ngokudandatheka. Kusenokwenzeka bafihla iimpawu zayo.
yedosi olusebenzayo ekhuselekileyo "Relaksona" abantwana nabo bakwishumi elivisayo abangaphantsi kweminyaka eli-18 ubudala iye ayasekwa ziingcali. Ngoko ke, ukuba ichiza kweli phakade akuvumelekanga.
Ngenxa iimpawu amayeza of a thile, oko kuchaphazela kakubi ukukwazi lomguli ukuqhuba izithuthi, kwakunye deal with imisebenzi enobungozi zifuna ukwandisa ingqalelo kunye nempendulo ngokukhawuleza. Kulo mba, ixesha unyango kunye eli chiza kufuneka silumke kakhulu.
Sleeping iipilisi "Relakson": nexabiso kunye analogue
Ichiza na indawo "Relakson"? Eli chiza, kukho ezikhethekileyo abaninzi. Ngempumelelo kakhulu amayeza zilandelayo: "Milovan", "imovan", "Thorson", "Somnol", "Slipvell", "Zolinoks", "Piklodorm", ". Zopiclone"
Zonke ezi machiza, kuquka "Relakson", sakhululwa kuphela ngokumiselwa ezikhemisti. Njengoko ngexabiso, ngoko ke kuthathwa kuthetha nga phezulu kakhulu. tablets 20 drug thile (7.5 mg) zakufumaneka 120-160 engange.
Izimvo ipilisi zokulala
Ngokutsho ubugcisa, iziyobisi "Relakson" imele besesithathu isizukulwana thile. Hi ndlela leyi, ezi ziquka i "Zaleplon" ne "zolpidem". La machiza kakuhle kakhulu kwaye ekhuselekileyo ngokupheleleyo.
Izigulane ingxelo yokuba emva kokuthatha iipilisi belele kakhulu siyiphuculeyo umgangatho ubuthongo. Nangona ngokupheleleyo ilondoloza ukulala bystrofazovy ezifunekayo ukuze kubuyiselwe imeko engqondweni nasemoyeni.
amayeza kujongwa inempembelelo omhle kade-yomtshangatshangiso kwisigaba ubuthongo, nto kubalulekile ukuba ukumimitheka ebonakalayo emzimbeni womntu.
Ngokutsho ubugcisa, kubelula iziyobisi esebenzayo normalizing iipateni balala na iintlobo ukuphazamiseka. Noko ke, yena okuba mncinane likhoboka.
Baqinisekiswa zibonisa ukuba ipilisi yokulala "Relakson 'Wanyamezela kakuhle kakuhle, kwaye alunasiphumo kwi kumsebenzi wemihla ngemihla woMntu. Noko ke, oogqirha musa singacebisi ukuthatha eli iyeza ngokwakho. Isigulana kufuneka kusoloko udibane nogqirha kwaye ulandele yonke idosi bubulumko.
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