ZempiloAmalungiselelo

Drotaverina hydrochloride

Drotaverina hydrochloride inxulumene sisincoko zoxubo ukuba ukusebenza spasmolytic. umsebenzi wayo sibhekiswe esihlunwini kakuhle kwenkqubo amalungu, enzala kunye biliary yokucola ukutya, kwakunye nemithambo egudileyo umaleko kwezihlunu. Drotaverina hydrochloride (Nospanum), ukukhuthaza ukuthanjiswa ngongqameko izihlunu agudileyo, uyakwazi ukuphelisa cramping. Ngaphezu koko, eli chiza kuphucula ijwabu yesondlo ioksijini ngokuthi kwandiswe sayo olujikeleza. Drotaverina hydrochloride uyakwazi ukutshintsha of weseli inwebu nobonisa permeability. Le medicament kunciphisa umsebenzi enzymatic of phosphodiesterase, ikhuthaza iyavumelana (uniform) ukwandisa amanqanaba Camp kunye nokufunxwa kokuqala kweeseli calcium ion.

Drotaverina hydrochloride lubonakala nezinga eliphantsi kokubonisa kunye iiproteni plasma. Isikakhulu sibopha ukuthi beta Alpha-globulin, albumin. Phakathi imizuzu mane anantlanu mathandathu emva nolawulo ngomlomo isicelo plasma ubonisa xi kwincopho into esebenzayo. Isiqingatha-bomi ngokomyalelo iiyure ezingamashumi amabini anesibini. Kukhuthaza metabolites eziveliswe kakhulu yokuchama. Inxalenye kukhuthaza beziyobisi yenzeka iingqatha.

Medicament (ngohlobo lwe ngenaliti, yaye amacwecwe) lwanziwa kuphelisa iintlungu kunye nesimo yiSpasticity spasm cupping. Drotaverina hydrochloride ubonisa isilonda esiswini, cholecystitis, ukuqhina, yiSpasticity umyalezo, pyloric agudileyo izihlunu spasm kunye cardinal kakhulu esiswini card, Ngokuzimela, nephrolithiasis, proctitis, pyelitis kunye uretrolitiaze. Ichiza lisetyenziswa amahlaba wamathumbu okubangelwa iigesi kokulibazisa wenze yiSpasticity. Le medicament nayo ingasetyenziswa xa eqhuba uxilongo, kuquka holetsistografii. Drotaverine esiwabelwe vasodilatation ekuchongeni nemithambo aqaqambayo smooth umaleko weplishi yintloko spasm nasezimpahleni lobuchopho. ichiza isoloko isetyenziswa algodismenoree practice yamanina. Le medicament uyakwazi ukunqanda ukuphelisa izihlunu gingxi mde wesibeleko ngexa lokukhulelwa kunye kwimeko zisongele isisu. Kwakhona kubonisiwe kwixesha delivery spasmolysis kwaye uthathe ukubhengeza zesibeleko umqala kunye ezikwenza kokubeleka.

hydrochloride Drotaverina. Imiyalelo.

A ukulungiselela ngohlobo iipilisi kufuneka zithathwe ngomlomo. Tablets akufuneki ukuhlafunwa okanye nakhandiweyo, kufuneka kuginywa lonke, amanzi ngokwaneleyo. Ichiza komntu akuxhomekekanga ekuzithandeleni ngexesha lesidlo. Oyidlayo kunye nexesha unyango kumiselwa ngamnye ngugqirha khona.

Ukuba intsha (ngaphezu ilishumi linamibini) kunye abadala ukuba aphelise iintlungu yiSpasticity amisele iipilisi 1-2 (40-80 mg) kabini okanye kathathu ngemini.

Abantwana abangaphantsi kweminyaka elishumi yokulungiselela inikwa ngokungqinelana kunye nokuqeshwa kagqirha.

Le medicament ngohlobo lwe ngenaliti ilawulwa intramuscularly. Izigulana insufficiency kwezintso okanye hepatic, kungenza ukuqaliswa ichiza yegazi. Le ndlela isebenza kuphela emva zokwamkelwa ngokuxwesileyo yesigulana. Xa ukuphazamiseka neuropathy yegazi leyo ibangwa nemithambo kwezihlunu smooth spasm layer ukuba ulawulo olucothayo intraarterial.

Njengomgaqo, izigulane ukulunyamezela amayeza. Noko ke, kwezinye iimeko, kusenokubakho iziphumo ebezingalindelekanga. Umzekelo, izigulane zinokuba isicaphucaphu, isitulo kakuhle, ukugabha. Inokwenzeka, kunye CNS nengxaki, ezifana waphula uphaphama kunye imo lokuphumla (ubuthongo), intloko ebuhlungu, niphele. Kwakukho iimeko ukuphazamiseka kwenkqubo sentliziyo, sabonakala tachycardia, arrhythmias, ukuthoba uxinzelelo. Kwakhona Ukudumba kunokwenzeka ukuba isifo ngeempumlo, negazi, bronchospasm.

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