ZempiloAmalungiselelo

"Tsinarin": imiyalelo ukusetyenziswa, nabalingani real

blocker calcium channel ekuthiwa iqela owahlukeneyo iziyobisi ukuba ube mnye isimiso ukusebenza, kodwa zahluke kwezinye izakhiwo, kuquka kwikinetiki parameters, izicwili selectivity kunye ukusebenza ngomhla izinga intliziyo.

Umgaqo basic yokusebenza amayeza ezinjalo kukuba banako ukuze kuthintelwe kwii-Ca ion ukusuka isithuba extracellular zibe iimpahla yegazi kunye neeseli imisipha yenhliziyo nge amajelo calcium (ngokucotha). Oku kukhokelela iqapheleka inyathelo vasodilator.

Eyona ethandwayo calcium ochasene sisiyobisi "tsinarin". Imiyalelo yokusebenzisa, ixabiso, kunye nohlaziyo ukwakhiwa loo mali iya kuchazwe ngezantsi.

ifomu ukukhululwa, ukupakishwa, inkcazelo, ukubunjwa

"Tsinarin" iziyobisi, izimvo zazo HIV, oko ithunyelwa ngokohlobo biconvex, ngeenxa kunye namacwecwe ezimhlophe. okanye icandelo labo oyinhloko cinnarizine. Ngaphandle kwalo, sisincoko kweziyobisi yenziwa njengoko excipients povidone K25, lactose, starch ingqolowa, colloidal lesilicon dioxide kunye wemagniziyam stearate.

Oku kuthetha ukuba unako ukuthenga kwi iiseli nentaba.

iimpawu imveliso

ngokusetyenziswa "tsinarin" iziyobisi Guide ingxelo ukuba ochasene uyakhetha lamajelo calcium (ngokucotha). Oku kunciphisa ukuphuma Ca ion kwizisele yaye kunciphisa inani plasmolemma izibuko, kodwa uphucula isiphumo vasodilating le carbon dioxide kunye kunciphisa kwezihlunu le arterioles.

Ngokwenza ngqo ezityeni, ichiza kunciphisa kakhulu abasabela ngayo izondlo (norepinephrine, epinephrine, angiotensin, vasopressin, kunye dopamine). Kwakhona qaphela ukuba medicament koqwalaselo vasodilating kwiipropati, kuquka nxamnye izitya lobuchopho. Kulo mzekelo, oko alunasiphumo kwi uxinzelelo lwegazi.

Drug "tsinarin", ixabiso yayo zidweliswe ngezantsi, iyanda sho umsebenzi antihistamine, lunciphisa excitability ye izixhobo vestibular kwaye kunciphisa umoya okanye ubunzulu NS novelwano. Eli chiza ngempumelelo liziphatha ngokungathi insufficiency sokuqala cerebrovascular kunye ezigulo ezondeleyo. Abantu namaphephandaba kakuhle peripheral iphucula kwegazi liya zonke izicwili kunye namaziko. Kwakhona yindlela yokunciphisa viscosity wegazi, kwandisa luthambe le inwebu iiseli ezibomvu kunye nokumelana umsipha hypoxia.

Le kinetics beziyobisi

Yintoni kwikinetiki iimpawu ezendeleyo iziyobisi "tsinarin"? Imiyalelo Sebenzisa uthi ukuba le arhente yi resorbed emathunjini kunye nesisu. Xi Incopho plasma afunyenwe emva kweeyure ezintathu. Unxibelelwano kunye iiproteni plasma cinnarizine yi-91%. Ichiza umzimba ngokupheleleyo esibindini. Its nesiqingatha sexesha-ubomi iiyure ezine. Kubonakala amayeza kwi umchamo ngendle.

ubungqina

"Tsinarin" Drug kuboniswe ulwamkelo:

  • komqondo saka;
  • stroke kobuchopho;
  • ukuhlukumezeka cranial;
  • Iimeko post-stroke (kuqukwa ukopha stroke);
  • olujikeleza Encephalopathy;
  • ngokuba kinetoses prophylaxis (lwaselwandle okanye isifo umoya, kwakunye nangexesha gungqa);
  • izifo vestibular (kuquka isifo Meniere kaThixo, ukuduma, vertigo, nystagmus, ukugabha kunye isicaphucaphu imvelaphi labyrinthine);
  • migraine (ngokuba yokuthintela isifo);
  • ephula ejikeleza yoluvo.

Izimo ukuya kuthabatha amacwecwe

Kuphantsi kwaziphi iimeko apho kufuneka ingamiselwa ichiza "tsinarin"? Imiyalelo iingxelo zokusetyenziswa ukuba eli yeza ke contraindicated ku:

  • hypersensitivity;
  • yokumitha;
  • ibele.

Kufuneka kuqatshelwe ukuba ichiza emiselweyo isilumkiso izifo Parkinson kaThixo.

Drug "tsinarin": imiyalelo yokusebenzisa

amacwecwe Ukuthatha kufuneka ajongwe ngaphakathi, ekukhethwa ukuba emva kwesidlo.

Xa aphazamiseka, iyeza igazi ebuchotsheni yaphathwa isixa 25-50 mg kathathu ngemini, kunye nokuhamba kwegazi peripheral - kwi 50-75 mg kunye ubuninzi efanayo.

Xa izifo vestibular Kucetyiswa ukuba ukuthatha amachiza 25 mg kathathu ngemini. Xa kinetosis okanye ekuthiwa "kwindlela" izigulane isifo omdala elawulwa-25 mg kweziyobisi imizuzu engama-30 phambi kohambo. Ukuba kuyimfuneko, iyeza walunyukiswa ngokuphindaphindiweyo emva kweeyure ezi-6 (kwi-mali efanayo).

Ngokuba abantwana, eli chiza imiselwe kwi-mali ka 1/2 ithamo omdala.

Xa uvakalelo oluphezulu ukuya kunyango medicament iqala isiqingatha idosi chu kunyuka. Ikhosi ye unyango angahlala naphi na ukusuka kwiiveki 2-3 ukuya iinyanga eziliqela.

imiphumela emibi

Eli chiza ingenza abasabela ecaleni zilandelayo:

  • umlomo owomileyo, ukuqunjelwa, iintlungu epigastric, senyongo cholestatic;
  • ukozela, intloko, ukudinwa, yaye disorder extrapyramidal (umzekelo, ukwanda kwezihlunu, lafa kwamalungu omzimba, hypokinesia);
  • planus ulele, ukubila, lupus-ezifana syndrome, irhashalala;
  • imiphumela negazi, ukutyeba, kunciphisa umfutho wegazi.

Price, iholide analogue iziyobisi kunye nohlaziyo ngayo

Ukukhupha amayeza ngoweqela of blocker calcium channel, wenziwe ngokumiselwa kagqirha. Price of ichiza malunga 20-50 engange.

Ukuba kuyimfuneko, isixhobo na indawo iziyobisi "Vertizin", "Diziron", "Stugezin", "stugeron", "Tsinazin", "Tsinedil" "Cinnarizine" njalo njalo.

Uninzi abathengi ngokuthatha lo ochasene, bathi ukuba sisiyobisi kakuhle kakhulu kwaye ngempumelelo. Iipilisi "tsinarin" inceda kuphelisa iingxaki vestibular kunye ukuphazamiseka kwinkqubo igazi. Ukongeza, eli chiza nempembelelo entle emzimbeni womntu kunye uqaqanjelwa, sengqondo esixhalabisayo saka kunye neemeko post-stroke.

Kufuneka kwakhona uqaphele ukuba le arhente ingqalelo sisoloko sisenza ngayo icala. Ukuze kuthintelwe uphuhliso lwabo, kufuneka zilandele ngqo zonke iingcebiso ugqirha. Athathe ipilisi "tsinarin" ngokwengqiqo yaso eyodwa, kuya kuvumeleka. Kufuneka kumiselwe kuphela ngugqirha khona.

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