Zempilo, Amalungiselelo
Medicament 'iflegi', imiyalelo zokusetyenziswa, iindlela kunye balawule
Drug "yeflegi" nto antiprotozoal antibiotics. Wamkelwa iyeza ngohlobo amacwecwe bhanya-camera emhlophe. Amalungiselelo ibandakanya metronidazole - le into esebenzayo, nto leyo ebonisa iimpawu zayo ezisisiseko, kunye nezixhobo: wemagniziyam stearate, starch, ingqolowa, hypromellose, povidone K30.
Izenzo amayeza "iflegi" umyalelo ukulungiselela umisela umsebenzi yalo phezulu antibacterial, indlela amanyathelo isiyobisi ukuncitshiswa zengqo- eqela elithile metronidazole nge iiprothini zothutho intracellular, nto leyo ekugqibeleni ekhokelela ekufeni ezincinane. Metronidazole liveza umsebenzi omkhulu-gazi abaninzi, eli qela iquka Trichomonas vaginalis, Lamblia intestinalis, ka Giardia intestinalis ezinye nesibopho anaerobes. Anayenza umsebenzi ophezulu ichiza nxamnye aerobes kunye anaerobes facultative.
Phantse ngoko nangoko emva kokuba ulwamkelo kukho olupheleleyo Absorption "iflegi" beziyobisi, yemiyalezo ibonisa ukuba kukufakwa ichiza aluchaphazeli isidlo. Ayithandi ephakamileyo ithotyelwe iqatshelwe kwemiphunga, ulusu, wesibindi nezintso, neencindi amadlozi kunye cerebrospinal, ematheni, kwaye netuwa lobufazi. Metabolization metronidazole ngokusebenzisa igcwala kwenzeka esibindini, beziyobisi livela becala nomchamo (malunga nama-70%), ixesha lekhefu, ukuqala ulwamkelo ukuya kwimveliso lokugqibela iiyure ezili-12.
Phakathi ezibonisa ukuba ukusetyenziswa "iflegi" libhekisela isikhokelo ukulungiselela izifo ezosulelayo ezifana:
- itrichomoniasisi enzala;
- giardiasis;
- amebiasis;
- හසුරුව isiphathi nonspecific.
Uhlobo kunye Iziganeko abosulelwe zinokwahluka apha irejimeni idosi ixesha lolwamkelo esikolweni "yeflegi" beziyobisi. Amacwecwe 2-PC. amaxesha 3 ngosuku abadala kuthatha iiveki amebiasis. Xa giardiasis bufinyeziwe ukuya kwiintsuku ezi-5 kwi idosi yemihla ngemihla ye-1 g itrichomoniasisi (හසුරුව isiphathi, urethritis) kwabasetyhini, urethritis emadodeni - emacwecweni 2 kwisithuba sexesha ezilishumi.
Kwezinye iimeko, kuba unyango lwezifo enzala unyango emiselweyo ichiza vaginally nje suppository.
Iziphumo ezingalindelekanga kunokuzenza nzima unyango "iflegi" Isikhokelo ukulungiselela iqulethe ulwazi malunga wabonakala kunokwenzeka elibi kwicala:
- CNS kwenzeka intloko ebuhlungu kunye nesiyezi kwiimeko ezinqabileyo - isiphithiphithi, unditsho, nemibono.
- sokugaya inkqubo, isicaphucaphu kwaye ayifane ibonakale emlonyeni, incasa sisinyithi, urhudo, ukugabha, kunye anorexia.
Kukho iimeko angawodwa ziyabagulisa ngokohlobo pruritus kunye urticaria, leukopenia kwenzeka ingakumbi xa lwamachiza unyango ixesha elide. Ukuba uyayeka ukuthatha ichiza, iimpawu shwaka ngoko nangoko.
Izimo ukuba ukusetyenziswa kweziyobisi "iflegi" imiyalelo kusebenza:
- anda kuvelana metronidazole;
- ngethuba lokukhulelwa nokuncancisa (ngenxa Ukuqhela metronidazole ngobisi lwebele);
imiyalelo ethile Phakathi kufuneka kuqatshelwe ukurhoxiswa zokusela utywala ngexesha unyango, ulawulo olungqongqo lwe ifomula kwegazi. Ngenxa enokuba yeziphumo ebezingalindelekanga njengokuba nesiyezi kunye nentloko kucetyiswa ukuba ukubaleka ngethuba konyango kunye naziphi na iindlela zokuhamba.
De namhlanje, akukho iingcebiso zonyango kuvela libanda yamayeza "yeflegi", kwiimeko ezinjalo, oko kufana nomqondiso. Akuvunyelwe ngokungqongqo ukuthatha unyango kunye namayeza eziqulathe ethanol (kwakunye kunye notywala), oko kunokubangela isiphumo esifanayo ekufumaneni disulfiram (umkhuhlane omkhulu, tachycardia, kunye nokugabha).
Ukuthengiswa beziyobisi eziveliswa ezikhemisti ngokumiselwa, elona xesha lininzi yokugcina - eyi-5 kwi tmax 250.
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