ZempiloUkuyeka ukutshaya

Macwecwe ngokutshaya "varenicline": izimvo kunye nemiyalelo yokusebenzisa

Ingxaki ukuyeka ukutshaya kudala ingqalelo omnye kakhulu embi. Akukho nto itshintshileyo ngoku. Inani abatshayayo luyanda minyaka yonke. abalandeli umkhwa inicotine imisiwe ukuthenga umdiza eselula kakhulu. Xa abakwishumi elivisayo, isenzo eso ezinxulumene kwingqikelelo mdala. Kodwa ixesha siqhubeka, umzimba saphule kusetyenziswa, oko kwenziwa kuxhomekeke nicotine. Kwaye ngoko ke Ingxaki iqala ngo yempilo: ezingwevu ngebala, a ukhohlokhohlo owomileyo, imibimbi ngaphambi kwexesha kwabasetyhini. Ngelishwa, umonakalo yecuba ukuba umzimba wethu siqala ukuphumeza kakhulu emva kwexesha. Asingabo bonke ajike ukunika ngokwakho. Kwiimeko ezinjalo, uyakwazi ukubhenela kwiziyobisi. Umzekelo, khetha ipilisi ukutshaya "varenicline". Namhlanje, ithandwa. Bona isincomo ngoogqirha, abantu abadumileyo, abantu abaqhelekileyo. Kutheni? Ngaphezu bafanelwe ukubalulwa obunjalo? Makhe zama ukulungisa oku phandle kunye.

Yini owenza izibalo

izifundo abasisigxina yokuhlalisana kunye ukuhlola kubonisa mhaka isenokunganambitheki xa uyicinga. Ehlabathini lonke, inani kubantu abangamadoda yi-50%. A abafazi abatshayayo isusela ukusuka-10% ukuya kuma-50%. Nantso lukhulu. Phantse isiqingatha sabantu emhlabeni kukuba nkqi kwenicotine. Ngoko ke, ukuba iipilisi namhlanje efanelekileyo nxamnye "varenicline" ukutshaya. Eneneni, phantse ama-70% abantu abatshayayo, eqonda ukuba ikhohlakeleyo nicotine, efuna ukuyeka ukutshaya. Kodwa kwenzeka ukuba asingabo bonke, kodwa% 5 kuphela. Kwaye nkqu kumandla yokuthanda, nangona, kakhulu, banokudlala indima ephambili kwakho ukuqalisa indlela yokuphila esempilweni. Kodwa kuyimfuneko ukuze bakuthathele ingqalelo kwenye into. Nicotine akukho enamazinga ngaphantsi iziyobisi. Umzekelo, cocaine okanye heroin. Yaye le ndoda akusoloko kusenzeka ukuba bamelane ngokwabo, ngenxa yokuba kukho utshintsho kakhulu emzimbeni. Kwaye apha ifikile uncedo "varenicline" iipilisi ngokutshaya. Ngaba zisiza? Ukuphonononga bacebisa ekufezekiseni yifuna. Kodwa yintoni ebangela ukuba ukusebenza ichiza?

A amagama ambalwa kwi intshongo

Ukuze siphendule lo mbuzo, wena nje kufuneka ukuqonda izenzo indlela nicotine. Kwaye ngoko ke ungakhetha indlela ukujongana nayo. Umzekelo, amacwecwe likhoboka nicotine "varenicline".

Eyona nto kukuba ungene umzimba wethu, inicotine wenza receptors ethile ebuchotsheni. Ngenxa yoko, kwisithuba nje imizuzwana embalwa emva kokuba le ndoda kwabakhukhumeleyo umdiza, uqala ku titwa a ukuzwa emnandi. Bona ahlangene kwakhululwa kungena egazini xa hormone okhethekileyo. Oogqirha bathi oku dopamine, okanye "iihomoni iziyolo". Kodwa ke ngokuhamba kwexesha eyavela unciphisa, kwaye kwakhona lo utshayayo iqala ukuba ubuhlungu. Kukho imfuneko umdiza entsha, ukufumana inxalenye mnandi.

Imbali i "varenicline"

Njengoko ubona, kukho isangqa eqhubekayo. Oku kukhokelela kukuba malunga nezigidi ezi-3 abantu abafa ngenxa yokutshaya. La manani akufunekanga yaziswe. Izazinzulu ziye kudala kunzima ekufuneni iindlela kulisindisa ihlabathi ukusuka isibetho ugwayi. Yaye ngenkulungwane yokuqala yama-21, kwafunyanwa isisombululo. "Varenicline" Kwakukho iipilisi ngokutshaya. Adunyiswe icebo yabo bobabo kwiZiko Neurobiology ebizwa Pfizer. Kuyinto umsebenzi weziko - mna noJyoti Co - ngoovulindlela yaye liphuhlise ipilisi ukuze akuncede uyeke ukutshaya.

Njani "varenicline" icwecwe?

Ngoko kwakukho iipilisi "varenicline 'ukutshaya. Ngaba zisiza? Yintoni na icebo yezenzo zabo? Makhe siye emva ukuziphatha kwenicotine. Kubonakala ukuba ifuthe layo phezu receptors nga ivaliwe. Indlela ukukwenza oko? elula kakhulu. indawo ugwayi kufuneka uthathe enye into. Ke akayi kuba nako ukwenza imisebenzi yalo yaye kunempembelelo ekhuthazayo. Musa ukuhlala kwindawo enye, nicotine iyaphuma emzimbeni kwaye akubangeli kuye nawuphi na umonakalo.

Kungenxa icebo kwaye lithetha imibala kwinkampani Pfizer. It luchaphazela receptors ingqondo, ngokwenjenjalo ngokubuyisela nicotine. Ngenxa yoko, iimpembelelo izinto eziyingozi ivaliwe. Indoda ayilufumani na kanene ugwayi. Ngenxa yoko, waza wafuna amacwecwe Ukutshaya "varenicline". Ingxelo evela kwabo bantu sele ngubani awathatha, zibonisa ukuba ebudeni kutsala, banganeli musa naziphi na iimvakalelo, kodwa ngokuchasene noko, lifumana incasa elibi. Ngenxa yoko, ungakunqweneli ukutshaya yehliswe kakhulu. Kuncipha uba amandla umnqweno imisiwe umdiza.

Kodwa "varenicline" ipilisi ilifa omnye impahla luncedo. Bona bayakwazi ukunciphisa iimpawu ezithi zenzeke xa ukuyeka ukutshaya. Oko kukuthi, umntu onesifo ezincinane emzimbeni.

Yintoni na oogqirha bathi?

Phambi kokuqala unyango kunye nemveliso ezintsha, kulungile ukuphulaphula kwiingcali. ngokwenene Oogqirha baqonde amacwecwe ngokutshaya "varenicline". Izimvo oogqirha bathi le sixhobo kunceda kakhulu ukuze aphumelele ekulweni nicotine. Abantu abaninzi ingqalelo abatshayayo enzima, wahlukana nalo mkhwa ngaphandle kobunzima.

Ukuqinisekiswa amazwi abo ukhonza manani zehlabathi. Drug emva ulingo lwezonyango waya ezithengiswayo ngo-2006. It ngenkuthalo waqala ukwamkela abatshayayo kumazwe awahlukeneyo. Kulo nyaka, amacwecwe Ukutshaya "varenicline" wasebenzisa abantu 9000. Kwaye 2007 waba yimbalasane kwinkampani Pfizer. Ichiza, kuphuhliswa Dzhotamom Co., waphumelela Galen. Kwezonyango ngayo kulingana ngexabiso Nobel Prize.

Noko ke, nangona eli zokuqaphela ngamazwe, bonke oogqirha bathi malunga side effects ukuba kwenzeka xa efumana imali. Sagqiba ekubeni ukhethe iipilisi litshaye 'varenicline "? Imiyalelo uza kunibalisela ngemeko zonke iipropati yayo. Well ukutyelela ugqirha wakho ukuba adibane naye. A Utyelelo kugqirha oyaziyo malunga nempilo yakho yonke kukunceda ukuba uphephe izinto ezi- angazithandiyo ngexesha unyango.

Siza kuthetha okungakumbi 'varenicline "

Ngoko ke ndigqibe ukuyeka ukutshaya? "Varenicline" iipilisi kukunceda nawe nale. Ngapha koko, ukuba ziqulathe varenicline. Le into ebizwa ochasene ugwayi. Varenicline uyakwazi ukukhuthaza nezamkeli nicotinic. Kodwa ke, ngokungafaniyo uninzi inicotine, impembelelo ngazo engephi. Yena uyakwazi ukuphembelela indlela unoxanduva lokuqulunqa engaziva iziyolo Ngecuba sitshaye. Varenicline iibhloko nje oko. Ngenxa yoko, lo utshayayo angacingi naluphi na isiphumo zokuqinisa, kunye nemfuneko Ukuqaleka kwayo ngcembe kunciphisa. Ukongezelela, varenicline ekwaziyo ukuphungula uyeka evela ngoko nangoko xa ekungaphumelelini icuba.

okufihliweyo varenicline

Njengoko kuchaphazela thina varenicline, eziqulathe "varenicline" icwecwe? Guide unika inkcazelo eneenkcukacha malunga nalo mba.

  • Varenicline ako kakuhle egazini, eqinisekisa ukusebenza kwayo. Le xi eliphezulu kufikelelwe iiyure 3-4 emva ongaka.
  • Le nto iza kuphela ebuchotsheni. Oku nombala kusiwa emzimbeni.
  • Kuyaphawuleka ukuba varenicline phantse ayitshintshi ubume bawo kwaye ungangeni naziphi abasabela emzimbeni. 92% beziyobisi salawo ingatshintshwanga. Kwaye kuphela i-8% ashiya imizimba yethu ngohlobo metabolites.
  • izinto kukhuthaza lwenziwa malunga 24 iiyure. Oko kukuthi, emva kokuba imini isidumbu sakho asiyi kufunyanwa phambi varenicline.
  • Ukongeza, le mveliso ingasetyenziswa kunye namanye amayeza. zophononongo zibonise ukuba varenicline akanayo naziphi na iimpawu ezingalunganga kwi ukudibana kunye nezinye iziyobisi.
  • Kodwa ezithatha ichiza kwisiqalo kunxilwe ezinxilisayo kungakhokelela kubunzima neuropsychiatric. Amahlaba - enye neziphumo elula kwiimeko ezinjalo.
  • Poor ufumana varenicline kunye nezinye anti-ukutshaya. Umzekelo, kunye efanayo "Nicorette". Kwiimeko ezinjalo, uyakwazi kwandisa umngcipheko yeziphumo ebezingalindelekanga.

Izimo

abatshayayo Abaninzi baye babona ukukhanya ekupheleni kwetonela emva ayesebenzisa tablet ngokutshaya "varenicline". Uhlaziya ubungqina ngempumelelo yabo. Kodwa musa aye ekhemesti elikufutshane kuthenga iiphakheji eziliqela. Abayi kuba luncedo kuwe. Isibakala sokuba esi sixhobo kufuneka Izimo yayo.

  1. Kubhetele ukuba bashiye ukusetyenziswa kweziyobisi ngethuba lokukhulelwa zisanyisa.
  2. Kwakhona akukho Kucetyiswa ukuba basebenzise abantu abaye babe imbali ukuphazamiseka kwengqondo kuluhlu.
  3. Kwiimeko of hypersensitivity ukuya varenicline lweziyobisi kwi sicelo asiyi kuqwalaselwa.

Ukongeza, ukutshaya "varenicline" iipilisi kufuneka kuthathwe:

  1. Abantwana abaye bengekafiki kwiminyaka eli-18 ubudala.
  2. Abaqhubi pilot. Ekubeni ichiza inceda ukwehlisa ingqalelo.
  3. Abantu abaphangelayo enxulumene kunye neendlela ngqo. Isizathu kukuba ezi Izimo efanayo - kukungakwazi ingqalelo, kwaye ingqalelo kweminwe.

imiphumela emibi

Kufuneka balumke ukuthatha iipilisi ngokutshaya "varenicline". Reviews zangaphambili abatshayayo bacebisa ukuba ngexesha unyango abaziva ixhala ongaqondakaliyo, iveze. Kwakukho iimeko kaninzi ugwayi. Enyanisweni, zonke ezi mpawu akufuneki ukuba lukoyikise. Ngapha koko, ukuba ziqhelekile bonke ukuyeka ukutshaya, nkqu ngaphandle kokubhenela kwi ichiza. Ngamanye amaxesha ungabona uxinzelelo lwegazi oluphezulu, abafundi inimba. Kwakhona senzeko Kuyaqondakala ukuba kuyenzeka, kuyimfuneko ukuba yokuhlambulula umzimba kwenicotine. Nangona kunjalo, zikhona iziphumo ebezingalindelekanga ezimandundu. Umzekelo, ezifana:

  • Ukuncipha kuyabuya lafaka.
  • Tachycardia.
  • Ekweneni ulwimi okanye kwingqula.
  • aqaqambayo.
  • Ezingekho.
  • Ugabhe, okanye ilindle wamagazi.
  • Exacerbation zizifo ezahlukahlukeneyo, usulelo woyiswa rhoqo wentsholongwane egazini.

Kamsinya nje uphawula kwi iimpawu ezifanayo, kufuneka ngoko nangoko uyeka ezithatha ichiza aze adibane nogqirha. Ugqirha uya kukunceda ukuba ukunyenyisa idosi. Kusenokwenzeka kunciphisa nto. Uya kwandula kuba lula umzimba ukuze wayesebenzisa yokungabikho kwenicotine.

Ukusetyenziswa "varenicline" tablets

Inzuzo ephambili yale iyeza yinto yokuba akukho mfuneko ukuba ukuyeka ukutshaya esithubeni. Oku kuthetha ukuba umntu uxinezeleko kangako. Unakho ancame isigarethi ke, xa iza kudlula ngokupheleleyo kwikhosi yonke. Kodwa iingcali Siyaleza ukulibala malunga nomnqweno wokwenza i yobunzima kwisiqingatha sesibini unyango.

Kungcono pre-ukufumanisa ngokwabo umhla xa ugqiba ekubeni unikezele midiza. Zengqondo Sicebisa ngokukhetha lusuku olumiselwe nasiphi na isiganeko ebalulekileyo kuwe. Qala ezithatha ichiza inokuba kwiveki phambi komhla ekhethiweyo.

Zonke iipilisi "varenicline" zibaliwe. Inika lula engaphezulu ngokuvumela ukuba zula, nini kwaye yintoni uhlobo tablet Kungcono ukuthatha.

Umthamo kwirejimeni "varenicline"

Nje ufuna ukukhankanya ukuba ikhondo unyango yenziwa ziintsuku 84. Ngamanye amaxesha kwaye zibeka ikhondo olongezelelweyo ngexesha elifanayo (iiveki ezili-12). Ukuba ngenxa unyango zange iphumelele iziphumo ezinqwenelekayo, ugqirha wakho angamisela kwikhosi yesibini ephambili.

amacwecwe Ukuthatha na nangaliphi na ixesha, kungakhathaliseki ukuba ukutya. Ngaloo ndlela babe iglasi ezele ngamanzi. Leyo yindlela kuya ngcono ukuba zifunxwe ngumzimba.

Kukho nomthamo irejimeni ekhethekileyo:

  • Iintsuku zokuqala 3 uthatha 1 emhlophe ipilisi kanye ngemini.
  • Iintsuku 4 elandelayo ithamo inyuswe. Kuya kufuneka sisele 1 ipilisi emhlophe amaxesha 2 ngosuku. Ngeli xesha, kungakuhle ukunciphisa inani yecuba watshaya ngamnye ngosuku.
  • Kwiiveki 11 ezayo, wena udle 1 tablet blue kabini yonke imihla. Ngokuqhelekileyo, ngeli xesha umzimba sele zilungiswe ngokupheleleyo ichiza, iziphumo ebezingalindelekanga lifinyele. Ngeli xesha ke kuyimfuneko ukuba bayeke ukutshaya.
  • Ngethuba lekhosi ufuna ukusebenzisa iipilisi ezongezelelweyo oluhlaza kabini ngemini.

Xa kunjalo, ukuba ningoyiki mkhuba ngethuba unyango aziyi kupheliswa ngokupheleleyo, kusenokungabikho ngoko nangoko ukuthatha iipilisi, yaye ngokuthe ngcembe nokunciphisa ithamo varenicline. Ukongeza, le ndlela kunyango uyakwazi ukukhusela iimpawu ndlongo ityala ngokungeyomfuneko, sokulibala, ukudakumba, ukubona kwayo, ukuba yasuka bayayeka ukuthatha ichiza.

Abadala kunye izigulane kwezintso kakuhle kwaye umsebenzi hepatic, utshintsho ithamo kwi inani leemeko ayikho imfuneko. Noko ke, ukuba nemiphumela emibi kakhulu, kufuneka udibane nogqirha. Njengomgaqo, lunciphisa ithamo kwisiqingatha sesibini yonyango tablet enye ngosuku.

cebiso Professional: indlela ukuyeka ukutshaya

iisayikholojisti abaninzi bathi enoba ngempumelelo okanye ulonwabele ichiza, ibe namandla ekulweni ukutshaya. Apha kufanelekile ukuba phinda ubulumko abantu: "On" varenicline 'ithemba, kodwa abo asina. " Inyaniso kukuba ukuze kuphunyezwe iziphumo ezintle, kufuneka ube umnqweno wakho kunye nenkuthazo. Izifundo yokuhlalisana kubonisa ukuba unyango kakhulu yimpumelelo kwabo izigulane ziye nzulu wagqiba ekubeni ayeke ukutshaya.

Kwakhona kubalulekile kulo mzekelo kunye nenkxaso abamthandayo, oogxa, obaziyo. Ukuba umntu othile nawe uya atshaye icuba, unako ngokulula kwaphula. Ngoko kuyimfuneko ukunciphisa okanye uxoxe nabantu abanjalo ukuba ubuncinane, okanye ashiye ngamathuba eziqatyana zokutshaya ethile kude.

Khetha: "varenicline" okanye "Tabeks"

Phakathi "varenicline" analogs kuquka iziyobisi ezifana "Tabeks". Abaninzi bakhetha igama lakhe, ngokuba kutshiphu. Kodwa yolingo lwezonyango baye babonisa ukuba cytisine (ngokusekelwe elenziwe elinganayo ngexabiso) isebenza ngaphantsi ngendlela eyiyo kwe varenicline. Xa kusetyenziswa "varenicline" umntu Ukwehluleka icuba, yaye, njengoko umthetho, oko kubo imbuyekezo kungekho ngaphezulu. Le ndawo mihla nezinempumelelo. Kubalulekile kakhulu kuyo, kunjalo, kokukhona ebiza "Tabex".

Price iipakethe ezimbini, equlethe amacwecwe-11 ka-500 mg 14 amacwecwe mg 1 1300-1400 engange. Kuba 112 tablets mg 1 Ukuze kuni makabeke malunga 3200 engange. Kakade ke, iindleko ungahluka kwimimandla eyahlukeneyo.

Mhlawumbi omnye umntu "varenicline" iipilisi zibonakala zibiza kakhulu, kodwa kuyaziwa elide ukuba impilo yabo kubhetele ukuba ukusindisa.

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