ZempiloAmalungiselelo

Ichiza "Tizanil": imiyalelo ukusetyenziswa, analogs kunye nohlolo

"Tizanil" - a relaxant kwezihlunu, enika amanyathelo engundoqo. Ukunciphisa ithowuni ye izihlunu skeletal basebenzisa iziyobisi "Tizanil" ezibonisa zokusetyenziswa ezivumela, ukuba kuyimfuneko, ukuphelisa aqaqambayo ezibangelwa uphuhliso isifo luvo, isifo idiskhi sisiba mandundu, utyando okanye ukwenzakala. Ngaphandle lezithako tizanidine esebenzayo, lo medicament iquka la macandelo ezongezelelweyo. effect Auxiliary kungenxa kubukho lesilicon dioxide, stearic acid, microcrystalline neselulosi kunye monohydrate lactose.

isenzo amayeza "Tizanila"

Alpha2-adrenergic receptors angababulali emva kokufumana "Tizanil" lithetha. Ukubunjwa kuqulunqo nga ngempumelelo ukujongana amahlaba wayibona wabonakalaliswa kwaye ziba ngendlela ezingapheliyo, ogama imvelaphi ubuchopho okanye lialio. Le arhente inceda ukwehlisa ukumelana kwezihlunu ngexesha iintshukumo eyimpumelelo ukwandisa izishunqulelo esicalanye dystrophy.

Kukufakwa beziyobisi kwenzeka ngokukhawuleza. "Tizanil" imiyalelo zokusetyenziswa njengoko sisixhobo ako phantse ngokupheleleyo kwi sixa siphezulu ezifumaneka egazini imizuzu engama-60 emva kokungena lokugaya.

Lokugaya kwenzeka esibindini, lo bioavailability elungelelene-34% njengesibophelelo kwi protein plasma - 30%. Kuba isiqingatha ubomi kuthatha umlinganiselo weeyure ezintathu. Ichiza salawo ivela emzimbeni njengoko metabolites ikakhulu izintso, isahlulo ayo lisusiwe lomelele.

ubungqina

Kuthetha ukuba "Tizanil" zibonisa ukuba ukusetyenziswa zimi ngolu hlobo lulandelayo:

  • Spine izifo kunye aqaqambayo, leyo zikhatshwa buhlungu;
  • aqaqambayo kabuhlungu emva kotyando;
  • skeletal UKUQINA kwemisipha ngenxa yezifo luvo.

Izimo ekufumaneni "Tizanila"

Amayeza contraindicated ne hypersensitivity amacandelo yayo, ukuphazamiseka kwesibindi kunye nezintso, akuba libizwe. "Tizanil" umyalelo awuvumeli ukuba isicelo ngexesha sokukhulelwa umntwana kunye nencum emondla. Contraindication na unyango "fluvoxamine". Age ngaphantsi kweminyaka eli-18, kubhekisela nasekuzeni ukuya Izimo.

Xa insufficiency kwezintso, lo myalelo ivumela ukuba ukusetyenziswa kweziyobisi, kodwa balumke ngeyona ndlela. Kukwasebenza kwanjalo kuyo ukusetyenziswa ngokudibeneyo "Tizanila" kunye inhibitors CYP1A2 kunye nonyango ebantwini abadala.

Isicelo medicament balawule

Iyeza sithathwa ngomlomo. Ukuba injongo nokusetyenziswa ichiza ukuphelisa aqaqambayo buhlungu, kucetyiswa ukuba kusetyenziswe yedosi ukusukela kuma-2 ukuya ku-4 mg. Ithamo Kucetyiswa-arhente kufuneka kuthathwe kathathu ngemini. Ukuba imeko enzima, uvunyelwe ukudibanisa kuhlonyelwa ngakumbi 2-4 mg medicament "Tizanil". Amacwecwe ngokwesikhokelo isicelo ingasetyenziswa kwemisipha skeletal UKUQINA 6mg. Le idosi iphezulu ngemihla, ngelo lokuqala unyango kufuneka kungagqithwa. Ekunyangeni iimeko ezinjalo ikhutshwa phandle nomthamo ezintathu yonke imihla. Ukuqwalasela isithuba seentsuku 3-7, ithamo ukuba kancane kancane ngomyinge we-3 mg.

Kuba kangangoko, Ukuzisa kuvumelekile idosi yemihla ngemihla ukuya mg-24. Umthamo elilelona jikelele 12 mg okanye ngaphezulu, kodwa ayikwazi ngaphezu 36 mg. Ngaloo mihla kufuneka kwenziwe 3 okanye 4 ukwamkelwa lithetha "Tizanil". Imiyalelo zokusetyenziswa iqulethe iinkcukacha malunga nonyango kwezigulane insufficiency kwezintso. izigulane ezinjalo ekuqaleni emiselweyo ichiza zokusetyenziswa kanye ngosuku idosi ubuncinane esilingana 2 mg. Idosi ichanekile ngcembe ingatshintshwa nge abasabela ngayo isigulane. Ukuba ufuna ukwandisa umthamo, ukwandisa umthamo kakhulu kuqala, uze emva koko utshintshe linani.

imiphumela emibi

unyango lwexesha elide maxa wambi ehamba ngayo zenyanyekayo eziphilayo. Kulo mzekelo, baye bakwazi ukuba ngakumbi kuvela ucaca ngakumbi. Oku kusebenza ulwamkelo amathamo ezinkulu "Tizanil" iziyobisi. Imiyalelo yokusebenzisa Ngokutsho kwezi ziziphumo ebezingalindelekanga, njengoko sibangelwa phecana zesisu, ndiyitshise le inwebu kwiinwebu emlonyeni, ukuhla nkoka uxinzelelo lwegazi, ukudinwa, ukozela, isiyezi kunye nezinye iziganeko ezibi.

Ukuvela yeziphumo ebezingalindelekanga isizathu sokuba unyango kugqirha, leyo mhlawumbi ukunciphisa idosi okanye rhoxisa ichiza, endaweni yalo ngezinye iindlela. Xa iipilisi unyango "Tizanil" imiyalelo yosetyenziso kufuneka waphawula ukuba umngcipheko yeziphumo ebezingalindelekanga inciphisiwe.

imithi

Impefumlelwano olwahlukileyo lwamayeza - oku lulwazi olubaluleke kakhulu, ekufuneka ziqwalaselwe phambi kokuba unyango ukunciphisa amathuba neziphumo ebezingalindelekanga, ngaphandle kakubi umzimba uze unciphise umngcipheko ukusebenza unyango.

Yinto eyaziwayo ukuba ichiza "Tizanil" edibene ne "Fluvoxamine", kukhokelela ngokonakala zempilo. Xa concomitantly ngeziyobisi umfutho bakwazi ukuphuhlisa bradycardia kunye hypotension.

Ukuba zombini ethanol okanye luvo ndaza tablets "Tizanil" umyalelo kubonisa ukwanda ukulalisa, okuyinto Ilungiselelwe "Tizanilom". Nge ile yakhe zokucwangcisa ngomlomo ukuze buthathaka yokususwa isiqingatha.

imithi Ungatshintsha ukusebenza konyango. Nokusebenzisa ngaxeshanye iziyobisi eziliqela, ukuze nokukhuthaza ifuthe kwenye okanye zisidimaze. Yonke le igcwele imbonakalo reactions ezibi, libanda, abanakho isiphumo kuyimfuneko.

oyi

Phambi kokuqala unyango with "Tizanil" Iimpawu kunye Izimo kufuneka ifundwe ngenyameko.

Kubikwe kukuvela inguqu engentle kwi nezintso nomhlehlo wesibindi. Kodwa yonyango esekelwe ukuthatha amachiza umthamo we-12 mg okanye ngaphantsi, amatyala anjalo ezinqabileyo kakhulu.

Kucetyiswa ukuba umane iimvavanyo umsebenzi kwesibindi. Kwiinyanga zokuqala ezine - ngenyanga kanye. Kwiimeko apho amanqanaba AST kunye ALT ngaphaya amaxabiso eziqhelekileyo ngaphezu kwabo ngokubonakalayo, ufuna ukupheliswa ichiza.

Ezinye izigulane abathatha "Tizanil" (kubandakanywa analogs) angavela ukozela. Nangona kule meko, awunako inxaxheba kwimisebenzi efuna ingqalelo ukwanda kunye nendlela asabela ngokukhawuleza.

Ngenxa nokoyikiswa ukuvuthuluka isigulane ichiza na irhoxisiwe wavele, oko ishiyelwa yi ekunciphiseni idosi ngcembe.

Analogs "Tizanila"

Kumiselwe imiyalelo kwiziko "Tizanil" ukufunda ayisoloko ukuvumela ukuba usebenzise indlela yokuqala ngenxa ezithile Izimo. Amachiza kuyabiza kakhulu zezethu "tizanidine-Teva" yaye "Tizalud". La machiza kwakhona relaxants, kufumaneka azipilisi babe isithako efanayo esebenzayo.

Bokwenziwa kunye nezinye analogs. Umzekelo, unyango kunokuba "Mydocalm", "Teva-Tizanilom" Surdaludom MR "," Surdaludom ".

reviews

Izimvo "Tizanile" zahlukile, okt. To. Ichiza zingachaphazela izigulane ngenye indlela. Kodwa ubukhulu becala ke HIV. Esi sibonelelo baqalisa ukuprinta ixesha elide, kuba phezu yentengiso ixesha elide, abantu abaninzi baye bakwazi ukuqinisekisa ukusebenza kwayo. Kukho izimvo amabi ashiywe ngenxa yeziphumo ezibi ngenxa wayengabunyamezeli yeekhomponenti okanye ukusetyenziswa amathamo eliphezulu ekucetyiswa ukuba unyango "Tizanil" iziyobisi. izimvo ezakhayo eshiywe ngabantu abonwabileyo kunye yoko, kule nkqubo yonyango athobele idosi emiselwe ngugqirha, kwaye phantse akazange isaziso nanini na embi abasabela ngayo.

ichiza wayedla ukunyanga isifo disc sisiba mandundu. Ngenxa iimpawu zayo inyathelo ezihamba isifo shwaka ngokukhawuleza. Gqithisela ebuhlungu kunye iqolo, ngcono impilo jikelele. Ngamanye amaxesha kukho iziphumo ebezingalindelekanga ezincinane ezifana ukozela, kome na isifo somlomo, kodwa hlengiso eyiyo idosi okanye ukurhoxiswa beziyobisi nyamalala. Ezinye izigulane yondele Intili osteochondrosis, musani ukubacaphukisa radicular syndrome, angala "Tizanil" babuyela ukuhamba eqhelekileyo, ngoxa amanye amayeza azizange iziphumo ezinqwenelekayo.

Ichiza ayikho kuyisusa embi phezulu izihlunu ithoni, nto leyo eye yaba ngenxa zestrowuku. "Tizanil" kuphela xa kagqirha phambi ezibonisa ezifanelekileyo. Ukuba unyango kufuneka kunye isibindi zizifo umntu okhulileyo okanye isigulane, kubhetele ukuba esichengeni impilo kwaye ukhethe relaxant kwezihlunu eyahlukileyo, nayo leyo alwa kakuhle imisebenzi.

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