Zempilo, Amalungiselelo
Ichiza 'pipolfen'. Imiyalelo yokusebenzisa
Enye kakhulu ngempumelelo arhente anti-kukwalisa, ngokuqhelekileyo kusetyenziswa kwiminyaka yakutshanje - "pipolfen". Imiyalelo ukusetyenziswa apho kwibhokisi nganye ichiza, kungakhathaliseki enoba evela pellet okanye isisombululo ukuba ulawulo ngo / kwi / m. Dragees "Pulpofena" zifana neentlumayo kukho phezu ecwebezelayo ye umbala ukukhanya-blowu, ngaphandle ivumba. Inaliti transparent, ngokuqhelekileyo enemibala emihle, kodwa ngamanye amaxesha tinged oluhlaza, akukho ivumba.
Ngenxa yokuba iphakheji ngamnye kufuneka ichiza "imiyalelo pipolfen 'ukusetyenziswa, abantu banokufunda intshukumo amayeza olufanelekileyo lwechiza. Le into esebenzayo kweli chiza - promethazine. It is a yemvelaphi phenothiazine, oko luphawulwa umsebenzi eliphezulu antihistamine. Promethazine ngokukhawuleza nangempumelelo kuchaphazela inkqubo luvo: has a thile, sine antipsychotic, antiemetic nefuthe hypothermic, kodwa ethoba kwaye kunqanda hiccups.
Drug "pipolfen" livimbela (kodwa ukubeka ecaleni ngokupheleleyo) iziphumo ezibangelwa histamine, kuquka ukurhawuzelela kunye ezindlwini. inyathelo Anticholinergic kwabangela ukusebenza yokomisa phezu kwiinwebu ngeempumlo nangomlomo.
Action promethazine antiemetic indalo yabangela ukuhla excitability ye izixhobo vestibular, umphumo esembindini anticholinergic, Uyeke umsebenzi mibono kunye nefuthe ngqo inhibitory kwiindawo ezithile zale Oblongata Medulla.
okulalisa beziyobisi ngenxa yokuba promethazine abangaphangeliyo histamine-N-methyltransferase kunye neebhloko ezi receptors histaminergic engundoqo. Ngaphezu koko, promethazine kwaye zinokuyithintela receptors acetylcholine serotinovye kananjalo ngokuvuselela receptors Alpha-adrenergic, ngqo ukuphuphumala yashukunyiswa ye lokusekwa reticular le brainstem. ukusebenza Antipsychotic of promethazine buthathaka phenothiazines antipsychotic, ngokuba ngezigqeba zazo yamachiza zahlukile kakhulu. Kulo mba, lo gama ezithatha ichiza ngendlela therapeutically owabelwe ithamo, promethazine Akukho iziphumo eziyingozi kwi nemithambo yegazi.
Okuqhotyoshelwe ichiza "Pipolphenum" umyalelo kwi isicelo sikuvumela ukuba ubone ukuba iziphumo bezonyango beziyobisi ziqala ukuvela emva kwemizuzu-2 (ukuba ichiza nolwathi intramuscularly) okanye imizuzu emi-5 (xa ilawulwa yegazi). Isenzo ichiza luhleli-avareji iiyure ezi-5, kodwa ngamanye amaxesha ingahlala ukuya kwiiyure ezili-12.
Ifumaneka isethi kunye nemveliso "pipolfen" umyalelo yenza kube lula ukuba baqhelane ezibonisa ukuba ukusetyenziswa kweziyobisi:
- nayiphi na zokubonisa izifo kukwalisa, kuquka nokuthimliswa, urticaria, hay fever, ukugula serum, ukurhawuzelela, angioedema, conjunctivitis;
- ngexesha therapy adjuvant ngayo anaphylactic;
- ukuhlanza okanye isicaphucaphu zomzimba eyabangelwa okanye ukubonakala emva ukusebenza;
- kusetyenziswa sine kwi ngeposi okanye ithuba ipreoperative;
- ntlungu kwenzeka emva kotyando;
- ukususa okanye ukuthintela isiyezi kunye isicaphucaphu, ezenzeka ngexesha ukuhamba kwizithuthi.
Noko ke, simele sikhumbule ukuba kukho Izimo kwi "pipolfen" iziyobisi. umyalelo Isicelo ikuvumela ukuba ufunde kubo ngendlela efanelekileyo:
- iimeko lubonakala ngokuba ukudandatheka le CNS;
- ukugabha imvelaphi elingachazwanga, lwenzeke manqaphanqapha ebantwaneni;
- ukusetyenziswa Ngokuhambelana utywala, analgesics ezidakumbisayo, elele iziyobisi;
- Kwiinyanga zokuqala ezimbini zobomi;
- Ukukhulelwa zisanyisa;
- ukuvalwa glaucoma.
Kwezinye iimeko, xa uthatha le amayeza nemiphumela emibi. Maxa wambi libanda, iziyobisi "Pipolphenum" esinokubakho. Izimvo zabantu ukuthatha eli yeza ukuze ube olunye ulwazi oluluncedo Kwiimeko ezinjalo.
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