ZempiloAmalungiselelo

Drug 'Atenolol Nycomed'

Kuba iziyobisi "Atenolol Nycomed" kukho imichiza, kwaye ezingoonombini ngamazwe kunye igama "Atenolol". Xa ulwimi ekhemisi pharmacologists ngokokwakheka ichiza ivela njenge (RS) -4- (2-hydroxy -3- (isopropylamino) phenyl-acetamide. Amacwecwe "Atenolol" zimele oboevypuklye iipilisi kugalelwe of umbala omhlophe, baye imilo philisi. Umzimba eziphambili ezinikiweyo notch zahlukane kwelinye icala, kukho imiqondiso AV55 kunye AV57.

Enye tablet ngokuxhomekeke kwifom release iqulethe neemiligram atenolol amahlanu okanye ikhulu elinye. Njengoko components abancedisayo kusetyenziswa talc, gelatin, propylene ethers, titanium dioxide, nemagnesium stearate, ipromeloza 2910 (15sP), umbona starch, isodiyam lauryl sulfate, enzima wemagniziyam carbonate.

Medicine "Atenolol Nycomed" izenzo njenge beta1-uyakhetha (cardioselective) adrenoceptor arhente ivalela, inwebu umsebenzi ozinzileyo ayikho. Esi sixhobo kubonisa ukusebenza antianginal, antiarrhythmic iqinile. Kuyinto olukwazi kuthintele beta-adrenergic receptors zentliziyo, ukunciphisa ukuvuselela engabalulekanga besahlulo onovelwano kwinkqubo luvo yawo kunye catecholamines, leyo kujikeleziswa egazini. Medicine "Atenolol" ukusebenza ngomhla ekunciphiseni sinus ukuzenzekela, normalizes izinga intliziyo ngxi kwaye ngexesha umthambo. Oku omeleza inkqubo kunye excitation of contractility engabalulekanga, kwi AV-Uhanjiso isiphumo linyuke. Xa isicelo sayo kukho ukuhla kwemfuno ioksijini engabalulekanga. Kakuhle kuchaphazela ukusebenzisa amayeza ngendlela "Atenolol" xa lisibekele uxinzelelo lwegazi. Ukuzinziswa umfutho kwenzeka ekupheleni kweveki yesibini ulwamkelo.

Ukulungiselela "Atenolol Nycomed" phezu indlela lolwamkelo ngomlomo ekwaziyo wendele wokugaya komthamo 50-60% ye idosi elawulwa. Kwazona kwi nomchamo kunye nesiqingatha-ubomi iiyure 6-7. La maxesha e izigulane ongaboniyo kwezintso, kuxhomekeke izinga product glomerular.

Izinto ezibonisa ukuba ichiza "Atenolol Nycomed" kukho iintlobo lwegazi kunye tachyarrhythmias (kubandakanywa sinus). Sebenzisa amayeza kwaye arhente lokuthintela isifo angina.

Idosi yemihla ngemihla beziyobisi ukuba abadala ukunyanga angina kunye noxinzelelo lwegazi ifikelela 50-100 mg. Amacwecwe yokwamkelwa wenza ukuya ku amaxesha amabini ngemini ngenxa yesibakala sokuba idosi yemihla ngemihla mayingagqithi 200 mg. Ukuhlamba ichiza kufuneka ibe isixa amancinci amanzi.

Iyeza isetyenziswa ngokuhambelana ngqongqo iingcebiso gqirha khona. Self-iyeza ayivumelekanga. Ichiza "Atenolol Nycomed" lineziphumo ebezingalindelekanga. Nemithambo yegazi unako ukuphendula imbonakalo ukuphazamiseka bradycardia, AV-Uhanjiso, usenokuba iminqweno of paresthesia nasemilenzeni ezibandayo, kwezinye iimeko zibonakale iimpawu ukusilela kwentliziyo. wokugaya uyaxabana elingalunganga isicaphucaphu iziyobisi, ukuqhina, urhudo, umlomo owomileyo (kunqabile), inkqubo yonyango - uphuhliso kangangoko imeko hypoglycemic kwizigulane ukubandezeleka seswekile, inkqubo enzala - ukuhla kunokwenzeka amandla. CNS reactions elibi nga ha kombisa ku yintloko, isiyezi, zokulala, ukudakumba, ukuziva ukudinwa. Kwakhona reactions kunokwenzeka kukwalisa, ukurhawuzelela, kwaye bomvu. Amatyala yokukhulisa umbilo, ukuncitshiswa secretion ukukrazuka ulwelo kwabhalwa, isenzeko conjunctivitis.

Kwakhona, kukho iqela Izimo. Xa uluhlu lwabo kubandakanya amanqanaba ngabanye ukusilela esingapheliyo intliziyo, bradycardia, hypotension, uvakalelo awongezelelekileyo okufumana ichiza, kunye nabanye.

Gcina amayeza kwindawo eyomileyo, ikhuselwe ekukhanyeni, ukukhutshelwa ngaphandle abantwana. lobushushu Room ku-25 ° C. A chiza igcina iipropati yayo iminyaka emihlanu.

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